SCHEMBL7656844

SCHEMBL7656844

CC(C)Oc1ccc(C(=O)Nc2ccc3c(c2)C(C)(C)N(C)CC3)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.50
RORC P51449 1/20 0.48
TMPRSS2 O15393 1/20 0.43
MEN1 O00255 2/20 0.43
POLB P06746 2/20 0.43
KMT2A Q03164 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
LMNA P02545 2/20 0.43
S1PR1 P21453 2/20 0.43
S1PR3 Q99500 1/20 0.43
GAA P10253 1/20 0.43
MCL1 Q07820 1/20 0.43
MAPT P10636 5/20 0.43
KCNQ3 O43525 1/20 0.42
KCNQ2 O43526 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TP53 P04637 3/20 0.42
ATM Q13315 1/20 0.42
NPC1 O15118 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6293739 0.83 ROCK2 (0.69) ROCK2RORCTMPRSS2CYP3A4
SCHEMBL7993309 0.82 ROCK2 (0.52) ROCK2RORCTMPRSS2MEN1POLB
SCHEMBL7655629 0.80 ROCK2 (0.50) ROCK2RORCTMPRSS2MEN1POLB
SCHEMBL6293978 0.80 ROCK2 (0.56) ROCK2RORCTMPRSS2S1PR1S1PR3
SCHEMBL6295101 0.79 ROCK2 (0.57) ROCK2RORCTMPRSS2MEN1KMT2A
SCHEMBL7657907 0.78 MAPT (0.63) MEN1POLBKMT2ALMNAMAPT
SCHEMBL7979562 0.78 MAPT (0.50) ROCK2MEN1POLBKMT2AMAPT
SCHEMBL7653578 0.78 RORC (0.47) ROCK2RORCMEN1POLBKMT2A
SCHEMBL7661456 0.77 RORC (0.47) ROCK2RORCTMPRSS2MEN1POLB
SCHEMBL7007156 0.76 ROCK2 (0.48) ROCK2RORCTMPRSS2LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed