SCHEMBL7657404

SCHEMBL7657404

CCCn1c(=O)c2[nH]c(N3CCN(Cc4ccccc4)CC3)nc2n2nc(Cc3ccccc3)nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
MAPK1 P28482 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HTT P42858 1/20 0.46
ADORA1 P30542 5/20 0.46
GAA P10253 1/20 0.46
ADORA2B P29275 4/20 0.45
ADORA3 P0DMS8 2/20 0.44
ALDH1A1 P00352 4/20 0.44
USP2 O75604 3/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ADORA2A P29274 3/20 0.43
ATM Q13315 1/20 0.42
RAB9A P51151 1/20 0.41
GLA P06280 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7661252 0.89 ADORA1 (0.47) MEN1KMT2AADORA1ADORA2BADORA3
SCHEMBL7656833 0.88 KMT2A (0.50) TSHRMEN1KMT2AADORA1ADORA2B
SCHEMBL8560002 0.83 ADORA1 (0.58) MEN1KMT2AADORA1ADORA2BADORA3
SCHEMBL7001583 0.81 ADORA2A (0.49) MEN1KMT2AADORA2BADORA3ALDH1A1
SCHEMBL7670431 0.70 ADORA2B (0.54) TSHRMAPK1MEN1KMT2AADORA1
SCHEMBL8560750 0.69 PDE4A (0.52) ADORA1ADORA2BADORA3HSD17B10ADORA2A
SCHEMBL7659412 0.67 ADORA2B (0.45) TSHRMAPK1MEN1KMT2AADORA1
SCHEMBL7666682 0.67 ADORA3 (0.50) TSHRMEN1KMT2AADORA1ADORA2B
SCHEMBL836300 0.66 ADORA2B (0.55) TSHRMAPK1MEN1KMT2AADORA1
SCHEMBL7668670 0.66 ADORA2B (0.51) TSHRMAPK1MEN1KMT2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492377-B1 Imidazotriazolopyrimidines with adenosine-antagonistic activity BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed