SCHEMBL7658556

SCHEMBL7658556

N#CCNC(=O)[C@@H](CNC(=O)c1ccccc1)S(=O)(=O)Cc1ccccc1OC(F)F

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSL P07711 11/20 0.42
CTSS P25774 7/20 0.42
CTSB P07858 6/20 0.42
CTSK P43235 5/20 0.41
ITGAV P06756 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6737505 1.00 CTSL (0.42) CTSLCTSSCTSBCTSKITGAV
SCHEMBL7656140 0.89 ITGAV (0.48) CTSLCTSSCTSBCTSKITGAV
SCHEMBL6062021 0.87 PPARG (0.46) CTSLCTSSCTSBCTSKITGAV
SCHEMBL6740637 0.86 CTSL (0.46) CTSLCTSSCTSBCTSK
SCHEMBL7548432 0.86 SLC22A12 (0.36) CTSLCTSSCTSK
SCHEMBL7661877 0.84 CTSL (0.43) CTSLCTSSCTSBCTSK
SCHEMBL6742062 0.83 CTSL (0.45) CTSLCTSSCTSBCTSK
SCHEMBL6737451 0.83 ALDH1A1 (0.50) CTSLCTSSCTSBCTSKITGAV
SCHEMBL6740031 0.82 CTSL (0.46) CTSLCTSSCTSBCTSKITGAV
SCHEMBL6740731 0.82 CTSL (0.46) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492362-B1 Compounds and compositions as cathepsin S inhibitors AXYS PHARMACEUTICALS, INC. 2002-12-10 US disclosed