SCHEMBL76595

SCHEMBL76595

Cc1cccc(C(=O)C(NC(=O)c2cccc(C)c2C)C(C)(C)C)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 10/20 0.50
KCNK9 Q9NPC2 9/20 0.50
KCNH2 Q12809 1/20 0.43
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
ATM Q13315 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL76896 0.91 NPC1 (0.45) KCNK3KCNK9NPC1RAB9ASMN1; SMN2
SCHEMBL76387 0.88 KCNK3 (0.47) KCNK3KCNK9NPC1RAB9ASMN1; SMN2
SCHEMBL77944 0.86 RAB9A (0.45) KCNK3KCNK9NPC1RAB9ATAS1R3
SCHEMBL10227845 0.86 KCNK3 (0.54) KCNK3KCNK9NPC1RAB9A
SCHEMBL10227846 0.77 ABCB1 (0.59) KCNK3KCNK9NPC1RAB9A
SCHEMBL10227844 0.75 NPC1 (0.48) NPC1RAB9ASMN1; SMN2
SCHEMBL10718970 0.74 ABCB1 (0.45) KCNK3KCNK9HDAC8HDAC6NPC1
SCHEMBL5056927 0.74 ABCB1 (0.42) KCNK3KCNK9HDAC8HDAC6NPC1
SCHEMBL8772420 0.72 ABCB1 (0.67)
SCHEMBL25607328 0.70 NPC1 (0.51) NPC1RAB9ATAS1R3TAS1R1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129355-B2 Nuclear receptor-based inducible gene expression system; modulating the expression of a gene in a host cell by introducing into the host cell a gene expression modulation system and activating that system using 5-ethyl-2,3-dihydro-benzo[1,4]dioxine-6-carboxylic acid (1-benzoyl-cyclopentyl)-amide INTREXON CORPORATION (US) 2012-03-06 US disclosed