SCHEMBL7659743

SCHEMBL7659743

COCc1oc(-c2c3ccccc3nn2Cc2ccccc2)nc1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
SCN8A Q9UQD0 2/20 0.51
PDE5A O76074 5/20 0.43
CYP2D6 P10635 1/20 0.39
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MPO P05164 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
CASP3 P42574 1/20 0.36
NR1H3 Q13133 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
CNR1 P21554 1/20 0.36
ACHE P22303 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4428683 0.81 PDE5A (0.61) CYP1A2SCN8APDE5ACYP2D6KDM4E
SCHEMBL4427114 0.72 VDR (0.50) KDM4EGAAPPARD
SCHEMBL13865173 0.70 PDE5A (0.53) CYP1A2SCN8APDE5ACYP2D6KDM4E
SCHEMBL4494497 0.68 ALDH1A1 (0.53) CYP1A2SCN8AL3MBTL1KDM4EALDH1A1
SCHEMBL4424864 0.68 F2RL3 (0.52) CYP1A2SCN8APDE5ACYP2D6KDM4E
SCHEMBL27669290 0.68 L3MBTL1 (0.56) CYP1A2SCN8ACYP2D6L3MBTL1KDM4E
SCHEMBL4434101 0.67 BUB1 (0.45) PDE5A
SCHEMBL4429083 0.67 PDE5A (0.58) CYP1A2SCN8APDE5ACYP2D6KDM4E
SCHEMBL9833283 0.64 ALDH1A1 (0.54) KDM4EALDH1A1LMNAPPARD
SCHEMBL4479319 0.64 SMN1; SMN2 (0.52) CYP1A2SCN8AKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414009-B1 CARDIOVASCULAR DISORDERS; ANTICOAGULANTS BAYER AKTIENGESELLSCHAFT (DE) 2002-07-02 US disclosed