SCHEMBL7660403

SCHEMBL7660403

CCOC(=O)C1CN(C(=O)c2ccccc2)CCN1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.48
HPGD P15428 1/20 0.46
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 1/20 0.45
TSHR P16473 2/20 0.45
BLM P54132 1/20 0.45
GAA P10253 1/20 0.45
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA4 P22748 2/20 0.44
CA9 Q16790 2/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656754 0.86 SIGMAR1 (0.51) SIGMAR1HPGDALDH1A1CA1CA2
SCHEMBL2628902 0.81 SIGMAR1 (0.55) SIGMAR1HPGDALDH1A1KDM4EBLM
SCHEMBL27799875 0.81 SIGMAR1 (0.58) SIGMAR1HPGDALDH1A1KDM4ECA1
SCHEMBL27854131 0.81 SIGMAR1 (0.58) SIGMAR1HPGDALDH1A1KDM4ECA1
SCHEMBL3306996 0.81 MAPT (0.39) ALDH1A1KDM4ETSHRGAA
SCHEMBL12261946 0.81 ALDH1A1 (0.64) ALDH1A1GAAPOLB
SCHEMBL9781792 0.80 PKM (0.50) ALDH1A1GAAPOLB
SCHEMBL28278676 0.78 CA1 (0.57) SIGMAR1HPGDBLMCA1CA2
SCHEMBL7801902 0.78 L3MBTL1 (0.54) SIGMAR1ALDH1A1KDM4E
SCHEMBL1658469 0.77 KDM4E (0.46) HPGDALDH1A1KDM4ETSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6469006-B1 PARTICULARLY FOR TREATING HIV INFECTIONS BRISTOL-MYERS SQUIBB COMPANY 2002-10-22 US disclosed
EP-1105135-A4 ANTIVIRAL INDOLEOXOACETYL PIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2001-12-12 EP disclosed
CN-1320037-A Antiviral indoloxoacetylpiperazine derivatives BRISTOL MYERS SQUIBB CO (US) 2001-10-31 CN disclosed
EP-1105135-A1 ANTIVIRAL INDOLEOXOACETYL PIPERAZINE DERIVATIVES BRISTOL-MYERS SQUIBB COMPANY (US) 2001-06-13 EP disclosed
WO-2000076521-A1 ANTIVIRAL INDOLEOXOACETYL PIPERAZINE DERIVATIVES BRISTOL-MYERS SQUIBB COMPANY (US) 2000-12-21 WO disclosed