SCHEMBL7664837

SCHEMBL7664837

N#CC(C#N)=C1N(CCSCc2cccc(CN3CCCCC3)c2)CCN1C(=O)c1cccc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.48
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 1/20 0.37
DRD4 P21917 4/20 0.36
BCHE P06276 2/20 0.36
ACKR3 P25106 1/20 0.36
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7663832 0.84 HRH3 (0.66) HRH3
SCHEMBL7665528 0.82 HRH3 (0.46) HRH3ACKR3
SCHEMBL7667137 0.80 HRH3 (0.48) HRH3
SCHEMBL7658659 0.77 HRH3 (0.68) HRH3
SCHEMBL7669477 0.75 HRH3 (0.49) HRH3
SCHEMBL7666194 0.74 HRH3 (0.47) HRH3
SCHEMBL7655572 0.74 PRMT6 (0.38) HRH3MEN1KMT2APOLB
SCHEMBL7666593 0.73 HRH3 (0.71) HRH3
SCHEMBL7662367 0.73 HRH3 (0.38) HRH3
SCHEMBL7667123 0.72 HRH3 (0.45) HRH3MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6495569-B1 CHEMOKINE ANTAGONISTS; TREATING DISEASE ASSOCIATED WITH INFLAMMATION AND/OR PATHOGENIC LEUKOCYTE RECRUITMENT AND/OR ACTIVATION MILLENNIUM PHARMACEUTICALS, INC. 2002-12-17 US disclosed
WO-2002085862-A1 IMIDAZOLIDINE DERIVATIVES AS CHEMOKINE RECEPTOR MODULATORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-10-31 WO disclosed