SCHEMBL7667137

SCHEMBL7667137

N#CC(C#N)=C1N(CCCc2ccccc2)CCN1CCSCc1cccc(CN2CCCCC2)c1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.48
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MCHR1 Q99705 1/20 0.39
SIGMAR1 Q99720 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7663832 0.84 HRH3 (0.66) HRH3
SCHEMBL7666194 0.82 HRH3 (0.47) HRH3ALDH1A1CYP2D6CYP2C9HIF1A
SCHEMBL7664837 0.80 HRH3 (0.48) HRH3
SCHEMBL7669477 0.80 HRH3 (0.49) HRH3
SCHEMBL7667123 0.80 HRH3 (0.45) HRH3
SCHEMBL7665528 0.79 HRH3 (0.46) HRH3
SCHEMBL7655572 0.78 PRMT6 (0.38) HRH3KDM4EALDH1A1CYP2D6CYP2C9
SCHEMBL7658659 0.76 HRH3 (0.68) HRH3
SCHEMBL7662367 0.76 HRH3 (0.38) HRH3CYP2D6CYP2C9HIF1A
SCHEMBL10668832 0.74 PRMT6 (0.50) HRH3KDM4EALDH1A1CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6495569-B1 CHEMOKINE ANTAGONISTS; TREATING DISEASE ASSOCIATED WITH INFLAMMATION AND/OR PATHOGENIC LEUKOCYTE RECRUITMENT AND/OR ACTIVATION MILLENNIUM PHARMACEUTICALS, INC. 2002-12-17 US disclosed