SCHEMBL7664864

SCHEMBL7664864

O=C(CC(F)(F)F)ON1CCC(CCS(=O)(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.43
ARG1 P05089 1/20 0.42
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
MAPT P10636 2/20 0.37
CA2 P00918 1/20 0.37
EIF4H Q15056 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
RORC P51449 1/20 0.35
AOC2 O75106 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5764628 0.87 HTR2A (0.43) CCR5ARG1HTR2AHTR2CCYP3A4
SCHEMBL7664869 0.74 CCR5 (0.40) CCR5ARG1NPC1RAB9A
SCHEMBL7607099 0.74 GPR119 (0.57)
Trifluoroacetic Acid SCHEMBL5764625 0.70 HSD11B1 (0.40) CCR5ARG1NPC1RAB9A
SCHEMBL6011594 0.69 CRBN (0.46) CCR5HTR2AHTR2CCYP3A4CYP2C19
Hydrochloric Acid SCHEMBL5763987 0.68 CRBN (0.45) HTR2AHTR2CCYP3A4CYP2C19
SCHEMBL19994599 0.67 MAOB (0.51) HTR2AHTR2C
SCHEMBL6011652 0.66 SLC6A4 (0.62) CCR5
SCHEMBL6011653 0.66 SLC6A4 (0.62) CCR5
SCHEMBL7734278 0.65 DRD2 (0.46) HTR2AHTR2CNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6498161-B1 TREATING INFECTION BY HIV; DELAYING OF THE ONSET OF AIDS; ASTHMA, ALLERGIC RHINITIS, DERMATITIS, CONJUNCTIVITIS, ATHEROSCLEROSIS OR RHEUMATOID ARTHRITIS MERCK & CO., INC. 2002-12-24 US disclosed