SCHEMBL7666259

SCHEMBL7666259

NC(=O)c1c[nH]nc1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
LMNA P02545 1/20 0.47
BCAT2 O15382 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.45
BRD4 O60885 1/20 0.42
IKBKB O14920 3/20 0.42
PARP1 P09874 3/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
CASP1 P29466 1/20 0.41
CDC7 O00311 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CCNA1 P78396 1/20 0.41
ALOX15 P16050 1/20 0.41
DHODH Q02127 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28034854 0.88 SCN9A (0.52) DHODHCTNNB1
SCHEMBL415485 0.85 KDM4E (0.55) KDM4ELMNASMN1; SMN2ALDH1A1ALOX15
SCHEMBL7729548 0.85 KDM4E (0.50) KDM4ELMNASMN1; SMN2MEN1KMT2A
SCHEMBL28304286 0.83 MAPK1 (0.44) LMNASMN1; SMN2IKBKBPARP1MEN1
SCHEMBL28460414 0.82 MKNK1 (0.51) PARP1DHODHSIRT1
SCHEMBL11957361 0.82 SMN1; SMN2 (0.49) KDM4ELMNASMN1; SMN2ALDH1A1GAA
Ethylene SCHEMBL27448159 0.82 KDM4E (0.51) KDM4ELMNASMN1; SMN2ALDH1A1ALOX15
SCHEMBL19663968 0.81 MAPK1 (0.56) KDM4ELMNAALDH1A1GAAALOX15
Biphenyl SCHEMBL895843 0.81 BCAT2 (0.46) KDM4EBCAT2BRD4IKBKBPARP1
SCHEMBL8913939 0.79 KDM4E (0.45) KDM4ELMNASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110023304-A Calpain regulator and its therapeutical uses 布莱德治疗公司 2019-07-16 CN disclosed
CN-109970654-A A series of substitution 2- phenylpyrazole derivatives and its preparation method and application 郑州大学 2019-07-05 CN disclosed
CN-105008344-B Bruton's tyrosine kinase inhibitor 辉瑞公司 2017-07-25 CN disclosed
CN-105008344-A Bruton's tyrosine kinase inhibitors PFIZER 2015-10-28 CN disclosed
US-6414013-B1 KINASE INHIBITORS; ANTICANCER AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2002-07-02 US disclosed