SCHEMBL7667245

SCHEMBL7667245

CC1CN(C(=O)Cn2c(=O)n(C)c3nc(-c4ccccc4)ncc32)CC(C)O1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 11/20 0.49
GRIN2B Q13224 11/20 0.49
TSPO P30536 1/20 0.48
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7210797 0.82 TSPO (0.57) GRIN1GRIN2BTSPO
SCHEMBL7217070 0.78 TSPO (0.53) GRIN1GRIN2BTSPOTSHRPOLB
SCHEMBL7216925 0.76 TSPO (0.56) GRIN1GRIN2BTSPOTSHRSMN1; SMN2
SCHEMBL7212081 0.76 LMNA (0.60) TSPOTSHR
SCHEMBL7215601 0.76 TSPO (0.58) GRIN1GRIN2BTSPO
SCHEMBL6482823 0.74 TSPO (0.61) GRIN1GRIN2BTSPO
SCHEMBL7215395 0.74 TSPO (0.67) GRIN1GRIN2BTSPO
Hydrochloric Acid SCHEMBL7212073 0.73 TSPO (0.60) GRIN1GRIN2BTSPO
SCHEMBL7217013 0.73 TSPO (0.58) GRIN1GRIN2BTSPO
SCHEMBL7667254 0.72 ALDH1A1 (0.38) TSPOTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6372740-B1 NERVOUS SYSTEM DISORDERS, ANTIEPILEPTIC AGENTS AND ANTIDEPRESSANTS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2002-04-16 US disclosed
EP-1036794-A1 2-ARYL-8-OXODIHYDROPURINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, MEDICINAL COMPOSITIONS CONTAINING THE SAME, AND INTERMEDIATES THEREOF Dainippon Pharmaceutical Co., Ltd. (JP) 2000-09-20 EP disclosed