SCHEMBL7672863

SCHEMBL7672863

CCCCCCn1cnc2c(OC)nc(Nc3ccccc3)nc21

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 7/20 0.52
CCNE1 P24864 7/20 0.52
CDK2 P24941 7/20 0.52
TK1 P04183 1/20 0.44
KCNH3 Q9ULD8 1/20 0.43
TMIGD3 P0DMS9 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
TAAR1 Q96RJ0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7661515 0.96 CCNE1 (0.54) PDGFRACCNE1CDK2TK1TMIGD3
SCHEMBL7668440 0.90 CCNE1 (0.51) PDGFRACCNE1CDK2TK1KCNH3
SCHEMBL7363250 0.88 TK1 (0.53) PDGFRACCNE1CDK2TK1TAAR1
SCHEMBL7661378 0.87 CCNE1 (0.51) PDGFRACCNE1CDK2TK1KCNH3
SCHEMBL7668634 0.87 CCNE1 (0.54) PDGFRACCNE1CDK2TK1TMIGD3
SCHEMBL7674300 0.86 CTSL (0.50) PDGFRACCNE1CDK2
SCHEMBL7667654 0.86 CCNE1 (0.53) PDGFRACCNE1CDK2TK1KCNH3
SCHEMBL7363934 0.85 CCNE1 (0.52) PDGFRACCNE1CDK2TK1TMIGD3
SCHEMBL7358873 0.85 CTSL (0.46) PDGFRACCNE1CDK2KCNH3
SCHEMBL24021926 0.84 CCNE1 (0.46) PDGFRACCNE1CDK2TMIGD3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414147-B1 DIAGNOSIS AND TREATMENT OF ANXIETY, DEPRESSION, SLEEP AND SEIZURE DISORDERS, DOWN'S SYNDROME, OVERDOSE WITH BENZODIAZEPINE DRUGS, AND FOR ENHANCEMENT OF MEMORY NEUROGEN CORPORATION 2002-07-02 US claimed
US-6414147-B1 DIAGNOSIS AND TREATMENT OF ANXIETY, DEPRESSION, SLEEP AND SEIZURE DISORDERS, DOWN'S SYNDROME, OVERDOSE WITH BENZODIAZEPINE DRUGS, AND FOR ENHANCEMENT OF MEMORY NEUROGEN CORPORATION 2002-07-02 US disclosed