SCHEMBL7674087

SCHEMBL7674087

COc1c(C#N)cccc1CO

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.41
ALDH1A1 P00352 2/20 0.41
IMPDH2 P12268 1/20 0.40
IMPDH1 P20839 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
GAA P10253 2/20 0.38
POLB P06746 1/20 0.38
HTR2A P28223 3/20 0.37
HTR2C P28335 1/20 0.37
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NPBWR1 P48145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20231243 0.84 TSHR (0.42) TSHRALDH1A1IMPDH2IMPDH1NPC1
SCHEMBL28252982 0.83 PTPN1 (0.36) TSHRALDH1A1IMPDH2IMPDH1NPC1
SCHEMBL16952177 0.83 ALDH1A1 (0.36) TSHRALDH1A1NPC1RAB9AGAA
SCHEMBL16953027 0.82 MAPT (0.35) TSHRALDH1A1NPC1RAB9AMAPT
SCHEMBL7717027 0.82 TSHR (0.38) TSHRALDH1A1IMPDH2IMPDH1NPC1
SCHEMBL7674083 0.82 TSHR (0.41) TSHRALDH1A1IMPDH2IMPDH1NPC1
SCHEMBL6736896 0.80 POLB (0.47) TSHRALDH1A1IMPDH2IMPDH1GAA
SCHEMBL129790 0.80 ALDH1A1 (0.46) ALDH1A1POLBMAPTSMN1; SMN2
SCHEMBL16956180 0.78 PDK2 (0.34) TSHRALDH1A1NPC1RAB9AMAPT
SCHEMBL23286532 0.76 IMPDH2 (0.38) ALDH1A1IMPDH2IMPDH1HTR2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900645-A1 3-PHENYLISOXAZOLIN DERIVATIVES WITH HERBICIDAL ACTION Bayer CropScience AG (DE) 2015-08-05 EP disclosed
US-6476021-B1 Compounds having cGMP-PDE inhibitory effect MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2002-11-05 US disclosed
EP-1048666-A1 NOVEL COMPOUNDS HAVING cGMP-PDE INHIBITORY EFFECT MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2000-11-02 EP disclosed