SCHEMBL7674433

SCHEMBL7674433

Cc1cc(C)c(-n2c3ccccc3c3c(N4CCC(N5CCCCC5)CC4)cc(C)nc32)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.41
CRHR1 P34998 1/20 0.40
HRH3 Q9Y5N1 5/20 0.37
EBP Q15125 1/20 0.36
DHCR7 Q9UBM7 1/20 0.36
CCR4 P51679 1/20 0.36
HSD17B10 Q99714 2/20 0.36
HPGD P15428 2/20 0.36
MAPK1 P28482 1/20 0.36
MBTD1 Q05BQ5 1/20 0.35
L3MBTL3 Q96JM7 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HTR1A P08908 1/20 0.35
ACVR1 Q04771 1/20 0.35
NPY2R P49146 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
KMT2A Q03164 1/20 0.35
PARP1 P09874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7679938 0.83 CRHR1 (0.47) NCF1CRHR1
SCHEMBL7677559 0.83 CRHR1 (0.45) NCF1CRHR1HSD17B10MAPK1HTR1A
SCHEMBL7679988 0.82 CRHR1 (0.43) NCF1CRHR1ACVR1
SCHEMBL7681552 0.82 NCF1 (0.52) NCF1CRHR1HSD17B10HPGDHTR1A
SCHEMBL7677542 0.81 CRHR1 (0.39) CRHR1
SCHEMBL7684787 0.80 NCF1 (0.55) NCF1CRHR1HTR1A
SCHEMBL7677573 0.80 CRHR1 (0.39) CRHR1
SCHEMBL7678166 0.77 CRHR1 (0.41) NCF1CRHR1HRH3HPGDL3MBTL1
SCHEMBL7684798 0.73 CRHR1 (0.51) CRHR1HSD17B10HPGDL3MBTL1KDM4E
SCHEMBL7674360 0.73 CRHR1 (0.39) CRHR1HPGDL3MBTL1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147085-A Aminoalkyl substituted 9H-pyridino[2,3-b] indole and 9H-pyrimidino[4,5-b] indole derivatives NEUROGEN CORPORATION (US) 2000-11-14 US claimed
US-6362186-B1 PSYCHOLOGICAL DISORDERS NEUROGEN CORPORATION 2002-03-26 US disclosed
US-6147085-A Aminoalkyl substituted 9H-pyridino[2,3-b] indole and 9H-pyrimidino[4,5-b] indole derivatives NEUROGEN CORPORATION (US) 2000-11-14 US disclosed