SCHEMBL7684787

SCHEMBL7684787

Cc1cc(C)c(-n2c3ccccc3c3c(N4CCCNCC4)cc(C)nc32)c(C)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 5/20 0.55
ADRB1 P08588 5/20 0.48
ADRB2 P07550 3/20 0.48
HTR1A P08908 7/20 0.42
HTR3A P46098 7/20 0.42
CRHR1 P34998 1/20 0.41
KDR P35968 1/20 0.39
HTR6 P50406 6/20 0.38
HTR2A P28223 4/20 0.38
HTR7 P34969 4/20 0.38
HTR2C P28335 3/20 0.38
HTR1D P28221 2/20 0.38
HTR2B P41595 2/20 0.38
HTR1B P28222 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
HRH2 P25021 2/20 0.36
SLC6A4 P31645 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7681552 0.96 NCF1 (0.52) NCF1ADRB1ADRB2HTR1AHTR3A
SCHEMBL7677559 0.84 CRHR1 (0.45) NCF1ADRB1ADRB2HTR1AHTR3A
SCHEMBL7674433 0.80 NCF1 (0.41) NCF1HTR1ACRHR1
SCHEMBL7682689 0.79 CRHR1 (0.51) NCF1ADRB1ADRB2HTR3ACRHR1
SCHEMBL7679938 0.79 CRHR1 (0.47) NCF1ADRB1ADRB2CRHR1
SCHEMBL7681555 0.78 NCF1 (0.44) NCF1ADRB1ADRB2HTR1AHTR3A
SCHEMBL7679988 0.78 CRHR1 (0.43) NCF1CRHR1HTR6HTR2B
SCHEMBL7677542 0.77 CRHR1 (0.39) CRHR1
SCHEMBL7677573 0.76 CRHR1 (0.39) CRHR1
SCHEMBL7076053 0.76 ADRB1 (0.39) NCF1ADRB1ADRB2HTR1AHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147085-A Aminoalkyl substituted 9H-pyridino[2,3-b] indole and 9H-pyrimidino[4,5-b] indole derivatives NEUROGEN CORPORATION (US) 2000-11-14 US claimed
US-6362186-B1 PSYCHOLOGICAL DISORDERS NEUROGEN CORPORATION 2002-03-26 US disclosed
US-6147085-A Aminoalkyl substituted 9H-pyridino[2,3-b] indole and 9H-pyrimidino[4,5-b] indole derivatives NEUROGEN CORPORATION (US) 2000-11-14 US disclosed