SCHEMBL767501

SCHEMBL767501

Nc1ccc2c(c1N)C(=O)NC2=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.50
THRB P10828 3/20 0.50
TDP1 Q9NUW8 3/20 0.50
MEN1 O00255 2/20 0.50
POLB P06746 2/20 0.50
MAPT P10636 2/20 0.50
APEX1 P27695 2/20 0.50
RECQL P46063 2/20 0.50
BLM P54132 2/20 0.50
KMT2A Q03164 2/20 0.50
CYP3A4 P08684 2/20 0.50
CASP7 P55210 2/20 0.50
RGS12 O14924 1/20 0.50
USP2 O75604 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
CASP1 P29466 1/20 0.50
BRCA1 P38398 1/20 0.50
MTOR P42345 1/20 0.50
GNAI1 P63096 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29260785 0.82 PARP1 (0.37) PARP1THRBTDP1MEN1POLB
SCHEMBL5171611 0.81 PARP1 (0.46) PARP1THRBTDP1MEN1POLB
SCHEMBL28982560 0.81 TDP1 (0.59) PARP1THRBTDP1MEN1POLB
SCHEMBL9450352 0.81 PPOX (0.48) PARP1THRBTDP1MEN1POLB
SCHEMBL7806624 0.78 PARP1 (0.47) PARP1THRBTDP1MEN1POLB
SCHEMBL7429649 0.78 THRB (0.55) PARP1THRBTDP1MEN1POLB
SCHEMBL10424885 0.77 PARP1 (0.42) PARP1THRBTDP1MEN1POLB
SCHEMBL5326248 0.77 PARP1 (0.39) PARP1THRBTDP1MEN1POLB
SCHEMBL6468586 0.77 PARP1 (0.50) PARP1THRBTDP1MEN1POLB
SCHEMBL29372946 0.76 PARP1 (0.53) PARP1THRBTDP1MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118271901-A Alcohol-soluble environment-friendly printing ink and preparation method thereof 厦门欧化实业有限公司 2024-07-02 CN claimed
EP-2373329-A2 USE OF EPIDERMAL GROWTH FACTOR INHIBITORS IN THE TREATMENT OF VIRAL INFECTION The Regents of the University of California (US) 2011-10-12 EP claimed
US-20110236349-A1 Use of Epidermal Growth Factor Inhibitors in the Treatment of Viral Infection THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2011-09-29 US claimed
WO-2010123527-A2 USE OF EPIDERMAL GROWTH FACTOR INHIBITORS IN THE TREATMENT OF VIRAL INFECTION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2010-10-28 WO claimed
WO-1997043643-A1 INHIBITORS OF PSEUDOMONAS AERUGINOSA INDUCED MUCIN PRODUCTION: COMPOSITIONS AND TREATMENTS FOR CYSTIC FIBROSIS PATIENTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-11-20 WO claimed
JP-5163240-A None JP disclosed
CN-118271901-A Alcohol-soluble environment-friendly printing ink and preparation method thereof 厦门欧化实业有限公司 2024-07-02 CN disclosed
EP-2066673-B1 TRICYCLIC COMPOUNDS AND ITS USE AS TYROSINE KINASE MODULATORS CHEMBRIDGE CORP (US) 2016-12-28 EP disclosed
US-9290503-B2 Tricyclic compound derivatives useful in the treatment of neoplastic diseases, inflammatory disorders and immunomodulatory disorders CHEMBRIDGE CORPORATION (US) 2016-03-22 US disclosed
US-9249147-B2 Tyrosine kinase inhibitors CHEMBRIDGE CORPORATION (US) 2016-02-02 US disclosed
EP-2966076-A1 NOVEL TYROSINE KINASE INHIBITORS ChemBridge Corporation (US) 2016-01-13 EP disclosed
CN-102036990-B Novel tyrosine kinase inhibitors CHEMBRIDGE CORP. (US) 2015-09-30 CN disclosed
CN-1102643-A Substituted derivatives of diaminophthalimide CIBA GEIGY AG (CH) 1995-05-17 CN disclosed
CN-1102643-A Substituted derivatives of diaminophthalimide CIBA GEIGY AG (CH) 1995-05-17 CN disclosed
EP-0516588-B1 Substituted diaminophtalimides and analogues CIBA GEIGY AG (CH) 1994-07-13 EP disclosed
EP-0600830-A1 Substituted derivatives of diaminophthalimide as protein-tyrosine kinase inhibitors CIBA-GEIGY AG (CH) 1994-06-08 EP disclosed
JP-H05163240-A SUBSTITUTED DIAMINOPHTHALIMIDE AND ANALOGUE CIBA GEIGY AG 1993-06-29 JP disclosed
CN-1067052-A The diaminophthalimides and the analogue thereof that replace CIBA GEIGY AG (CH) 1992-12-16 CN disclosed
CN-1067052-A The diaminophthalimides and the analogue thereof that replace CIBA GEIGY AG (CH) 1992-12-16 CN disclosed
EP-0516588-A1 Substituted diaminophtalimides and analogues CIBA-GEIGY AG (CH) 1992-12-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110236349-A1 Use of Epidermal Growth Factor Inhibitors in the Treatment of Viral Infection EGFR, HDGF, HGF PARP1 4324/4885THRB 819/4885TDP1 3634/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.