SCHEMBL7677576

SCHEMBL7677576

Cc1cc(C)c(-n2c3ccccc3c3c(C4CCCN4NC4CCCC4)cc(C)nc32)c(C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 2/20 0.39
NPY1R P25929 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 3/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
NPC1 O15118 1/20 0.32
NR2F2 P24468 1/20 0.32
LMNA P02545 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HCRTR1 O43613 1/20 0.30
POLB P06746 1/20 0.30
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674366 0.86 CRHR1 (0.40) CRHR1NPY1RKDM4EALDH1A1GAA
SCHEMBL7675196 0.86 CRHR1 (0.40) CRHR1NPY1RKDM4EALDH1A1GAA
SCHEMBL7677573 0.74 CRHR1 (0.39) CRHR1
SCHEMBL7677887 0.74 CRHR1 (0.45) CRHR1KDM4EALDH1A1GAARAB9A
SCHEMBL7674360 0.74 CRHR1 (0.39) CRHR1NPY1RKDM4EALDH1A1GAA
SCHEMBL7675191 0.74 CRHR1 (0.39) CRHR1NPY1RKDM4EALDH1A1GAA
SCHEMBL7677542 0.72 CRHR1 (0.39) CRHR1
SCHEMBL7674433 0.71 NCF1 (0.41) CRHR1KDM4EALDH1A1KMT2A
SCHEMBL7684798 0.71 CRHR1 (0.51) CRHR1KDM4EALDH1A1GAALMNA
SCHEMBL7788898 0.70 CRHR1 (0.48) CRHR1NPY1RKDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147085-A Aminoalkyl substituted 9H-pyridino[2,3-b] indole and 9H-pyrimidino[4,5-b] indole derivatives NEUROGEN CORPORATION (US) 2000-11-14 US claimed
US-6362186-B1 PSYCHOLOGICAL DISORDERS NEUROGEN CORPORATION 2002-03-26 US disclosed
US-6147085-A Aminoalkyl substituted 9H-pyridino[2,3-b] indole and 9H-pyrimidino[4,5-b] indole derivatives NEUROGEN CORPORATION (US) 2000-11-14 US disclosed