SCHEMBL7678632

SCHEMBL7678632

CCC(=O)N(CCN1CCOCC1)c1c[nH]c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 2/20 0.50
CHRM3 P20309 1/20 0.47
CYP2D6 P10635 1/20 0.47
HTR2A P28223 4/20 0.45
HTR7 P34969 4/20 0.45
DRD2 P14416 2/20 0.45
OPRM1 P35372 2/20 0.45
SIGMAR1 Q99720 1/20 0.45
KCNH2 Q12809 1/20 0.45
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
HRH3 Q9Y5N1 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
MITF O75030 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7671809 0.90 ALDH1A1 (0.48) CYP2D6HTR2AHTR7DRD2OPRM1
SCHEMBL7677414 0.88 OPRM1 (0.46) CYP2D6HTR2AHTR7DRD2OPRM1
SCHEMBL7678792 0.82 ALDH1A1 (0.47) HTR2AHTR7DRD2KCNH2ALDH1A1
SCHEMBL7675804 0.76 HTR6 (0.55) HTR2AHTR7DRD2KCNH2
SCHEMBL13763428 0.76 TACR2 (0.57) TACR2CHRM3CYP2D6ALDH1A1KDM4E
SCHEMBL7677881 0.76 HTR1A (0.57) CYP2D6HTR2AHTR7ALDH1A1CYP1A2
SCHEMBL7677363 0.73 NPSR1 (0.54) ALDH1A1KDM4ELMNAKMT2AMEN1
SCHEMBL13757476 0.73 TACR2 (0.54) TACR2CHRM3CYP2D6HTR2AHTR7
SCHEMBL7839785 0.73 OPRM1 (0.48) OPRM1SIGMAR1ALDH1A1LMNACYP2C19
SCHEMBL29336734 0.71 CYP2D6 (0.48) TACR2CHRM3CYP2D6HTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472418-B1 Non-peptide NK1 receptors antagonists WARNER-LAMBERT COMPANY 2002-10-29 US disclosed