SCHEMBL7680090

SCHEMBL7680090

COC(=O)CC(C[N+](=O)[O-])c1cccc(Cl)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
ALDH1A1 P00352 5/20 0.36
GAA P10253 1/20 0.36
CYP3A4 P08684 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
NFKB1 P19838 1/20 0.36
PNMT P11086 1/20 0.36
CACNA2D1 P54289 2/20 0.35
CACNA1B Q00975 2/20 0.35
CACNB1 Q02641 2/20 0.35
CACNA1G O43497 1/20 0.35
LMNA P02545 1/20 0.35
GLA P06280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6487215 0.90 ALDH1A1 (0.42) ALDH1A1GAACYP3A4LMNA
SCHEMBL6487800 0.85 CNR1 (0.38) MEN1KMT2ATAS1R3TAS1R1TAS1R2
SCHEMBL6479396 0.82 L3MBTL1 (0.36) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL6479354 0.81 MAPT (0.39) MEN1KMT2AMAPTALDH1A1GAA
SCHEMBL7684336 0.80 ALDH1A1 (0.40) POLBMAPTALDH1A1GAACYP3A4
SCHEMBL7687237 0.80 CNR1 (0.43) MAPTALDH1A1CYP3A4
SCHEMBL7431251 0.80 MAPT (0.45) MEN1KMT2AMAPT
SCHEMBL7686449 0.80 CYP2C19 (0.41) MEN1KMT2AMAPTALDH1A1CYP1A2
SCHEMBL6477248 0.79 CYP2C9 (0.45) KMT2AMAPTALDH1A1CYP3A4LMNA
SCHEMBL6492632 0.79 ALDH1A1 (0.40) POLBMAPTALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492392-B1 INHIBITING TUMOR CELL PROLIFERATION KYOWA HAKKO KOGYO CO., LTD. (JP) 2002-12-10 US disclosed
WO-2001085716-A1 2-PIPERIDONE COMPOUNDS FOR THE TREATMENT OF CANCER KYOWA HAKKO KOGYO CO., LTD (JP) 2001-11-15 WO disclosed