SCHEMBL7680358

SCHEMBL7680358

CCc1cccc2cccc([C]=O)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.47
GABRB2 P47870 4/20 0.47
ELANE P08246 6/20 0.38
CYP1B1 Q16678 2/20 0.35
NSD2 O96028 1/20 0.35
CASP6 P55212 1/20 0.35
GFER P55789 1/20 0.35
DAO P14920 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
HTR2A P28223 2/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KCNH2 Q12809 1/20 0.33
SCN5A Q14524 1/20 0.33
CASP1 P29466 1/20 0.33
MPI P34949 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15861173 0.82 CA1 (0.43) GABRA1GABRB2ELANETSHR
SCHEMBL6443578 0.80 ALDH1A1 (0.45) CYP1B1ALDH1A1HPGDCYP1A1CYP1A2
SCHEMBL3244580 0.80 GABRA1 (0.52) GABRA1GABRB2ELANECYP1B1NSD2
SCHEMBL10628200 0.78 CYP1A2 (0.43) DAOALDH1A1HTR2ACYP1A2CYP3A4
SCHEMBL535892 0.76 GABRA1 (0.45) GABRA1GABRB2ALDH1A1
SCHEMBL9849127 0.75 GABRA1 (0.45) GABRA1GABRB2DAOCYP3A4KCNH2
SCHEMBL1049567 0.75 GABRA1 (0.45) GABRA1GABRB2DAOCYP3A4KCNH2
SCHEMBL7680857 0.75 CYP1A2 (0.40) ELANECYP1B1ALDH1A1HPGDCYP1A1
SCHEMBL9670621 0.73 GABRA1 (0.44) GABRA1GABRB2DAOALDH1A1TSHR
SCHEMBL9099235 0.73 KDM4E (0.41) GABRA1GABRB2CYP1B1ALDH1A1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3743061-A1 CANNABINOIDS AND DERIVATIVES FOR PROMOTING IMMUNOGENICITY OF TUMOR AND INFECTED CELLS Pascal Biosciences Inc. (CA) 2020-12-02 EP claimed
WO-2019144126-A1 CANNABINOIDS AND DERIVATIVES FOR PROMOTING IMMUNOGENICITY OF TUMOR AND INFECTED CELLS PASCAL BIOSCIENCES INC. (CA) 2019-07-25 WO claimed
EP-3743061-A1 CANNABINOIDS AND DERIVATIVES FOR PROMOTING IMMUNOGENICITY OF TUMOR AND INFECTED CELLS Pascal Biosciences Inc. (CA) 2020-12-02 EP disclosed
WO-2019144126-A1 CANNABINOIDS AND DERIVATIVES FOR PROMOTING IMMUNOGENICITY OF TUMOR AND INFECTED CELLS PASCAL BIOSCIENCES INC. (CA) 2019-07-25 WO disclosed
US-6359148-B1 FOR POLYMER, LUBRICANTS; HEAT, OXIDATION RESISTANCE, PHOTOSTABILITY NESVADBA PETER (CH) 2002-03-19 US disclosed
US-6346630-B1 3-Arylbenzofuranones as stabilizers CIBA SPECIALTY CHEMICALS CORPORATION 2002-02-12 US disclosed
EP-0648765-B1 Process for the production of 3-arylbenzofuranones CIBA SC HOLDING AG (CH) 2000-07-12 EP disclosed
US-5814692-A PROTECTING POLYMERS AND LUBRICANTS AGAINST THERMAL, OXIDATIVE OR LIGHT-INDUCED DEGRADATION CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-09-29 US disclosed
US-5807505-A HEAT AND OXIDATION RESISTANCE, PHOTOSTABILITY OF POLYMERS CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-09-15 US disclosed
US-5773631-A PROTECTION OF POLYMERS AND LUBRICANTS AGAINST THERMAL, OXIDATIVE OR LIGHT INDUCED DEGRDATION CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-06-30 US disclosed
US-5693829-A PROTECT AGAINST THERMAL, OXIDATIVE OR LIGHT-INDUCED DEGRADATION CIBA SPECIALTY CHEMICALS CORPORATION (US) 1997-12-02 US disclosed
US-5614572-A Benzofuran-2-ones as stabilizers CIBA-GEIGY CORPORATION (US) 1997-03-25 US disclosed
US-5607624-A Process for the preparation of 3-arylbenzofuranones CIBA-GEIGY CORPORATION (US) 1997-03-04 US disclosed
US-5516920-A POLYMER STABILIZERS CIBA-GEIGY CORPORATION (US) 1996-05-14 US disclosed
EP-0648765-A1 Process for the production of 3-arylbenzofuranones CIBA-GEIGY AG (CH) 1995-04-19 EP disclosed