SCHEMBL7680461

SCHEMBL7680461

Cc1cc2c(cc(C(=O)O)n2Cc2ccc(F)c(Cl)c2)o1

nearest known ligand 0.81

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 2/20 0.81
MAPT P10636 7/20 0.60
LMNA P02545 1/20 0.56
CCR2 P41597 10/20 0.53
ALDH1A1 P00352 3/20 0.50
KDM4E B2RXH2 2/20 0.50
HPGD P15428 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
ALOX15 P16050 1/20 0.50
ALOX12 P18054 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HSD17B10 Q99714 1/20 0.50
TP53 P04637 1/20 0.49
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7680884 0.91 ABCB11 (0.81) ABCB11MAPTLMNACCR2ALDH1A1
SCHEMBL7691746 0.90 ABCB11 (1.00) ABCB11MAPTLMNACCR2
SCHEMBL7679796 0.88 MAPT (0.80) ABCB11MAPTLMNAALDH1A1KDM4E
SCHEMBL7701288 0.79 MAPT (0.76) ABCB11MAPTLMNAALDH1A1KDM4E
SCHEMBL7679941 0.77 ABCB11 (0.78) ABCB11CCR2
SCHEMBL7682546 0.76 ABCB11 (0.76) ABCB11MAPTLMNAALDH1A1KDM4E
SCHEMBL6598061 0.76 CCR2 (0.79) ABCB11CCR2
SCHEMBL7682571 0.75 ABCB11 (0.73) ABCB11CCR2
SCHEMBL7680085 0.74 ABCB11 (0.73) ABCB11CCR2
SCHEMBL6597871 0.74 CCR2 (0.80) ABCB11CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6479527-B1 Bicyclic pyrrole derivatives as MCP-1 inhibitors ASTRAZENECA UK LIMITED (GB) 2002-11-12 US disclosed