SCHEMBL7681304

SCHEMBL7681304

COc1ccc(F)cc1C1CC(=O)CC(=O)C1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.45
HTR2C P28335 4/20 0.45
HTR2B P41595 3/20 0.45
SLC6A2 P23975 4/20 0.44
SLC6A4 P31645 4/20 0.44
SLC6A3 Q01959 2/20 0.44
KDM4E B2RXH2 1/20 0.40
TSHR P16473 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
MAP1LC3B Q9GZQ8 1/20 0.40
TP53 P04637 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7679054 0.84 HTR2C (0.45) HTR2AHTR2CHTR2BSLC6A2SLC6A4
SCHEMBL7685135 0.81 TP53 (0.46) KDM4EPDE4APDE4BPDE4CPDE4D
SCHEMBL30368251 0.80 MAP1LC3B (0.57) HTR2CMAP1LC3BTP53RECQL
SCHEMBL643845 0.80 MAP1LC3B (0.57) HTR2CMAP1LC3BTP53RECQL
SCHEMBL21231846 0.80 SLC6A2 (0.54) HTR2AHTR2CHTR2BSLC6A2SLC6A4
SCHEMBL6794592 0.79 SLC9A1 (0.43) TP53RECQL
SCHEMBL29648490 0.78 CYP3A4 (0.46) HTR2AHTR2CKDM4EPDE4APDE4B
SCHEMBL6794027 0.78 KDM1A (0.46) TP53RECQL
SCHEMBL30472850 0.78 KDM4E (0.41) HTR2AHTR2CHTR2BKDM4EPDE4A
SCHEMBL2571867 0.77 PTGDR2 (0.56) HTR2AHTR2CHTR2BSLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed