SCHEMBL7685135

SCHEMBL7685135

COc1ccc(Cl)cc1C1CC(=O)CC(=O)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.46
RECQL P46063 1/20 0.46
ADAM17 P78536 1/20 0.43
PTGDR2 Q9Y5Y4 8/20 0.42
PTGDR Q13258 5/20 0.42
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11817691 0.88 TP53 (0.46) TP53RECQLADAM17PTGDR2PTGDR
SCHEMBL7681304 0.81 HTR2A (0.45) TP53RECQLKDM4EPDE4APDE4B
SCHEMBL7687548 0.79 TP53 (0.50) TP53RECQLPOLBMAPT
SCHEMBL7685246 0.79 TP53 (0.41) TP53ADAM17PTGDR2PTGDRALDH1A1
SCHEMBL29648490 0.78 CYP3A4 (0.46) TP53RECQLKDM4EPDE4APDE4B
SCHEMBL7685669 0.78 TP53 (0.62) TP53RECQLALDH1A1POLBMAPT
SCHEMBL30368545 0.77 TP53 (0.49) TP53RECQLALDH1A1KDM4EHPGD
SCHEMBL30368251 0.77 MAP1LC3B (0.57) TP53RECQLALDH1A1MAPT
SCHEMBL643845 0.77 MAP1LC3B (0.57) TP53RECQLALDH1A1MAPT
SCHEMBL7683113 0.77 TP53 (0.51) TP53RECQLPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed