SCHEMBL7681995

SCHEMBL7681995

O=C(c1ccccc1)c1ccc(C(C(=O)O)C(=O)O)c([N+](=O)[O-])c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.62
VCAM1 P19320 2/20 0.62
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
ALDH1A1 P00352 2/20 0.47
PDK1 Q15118 1/20 0.46
POLB P06746 1/20 0.45
CASP6 P55212 1/20 0.45
CDC25B P30305 1/20 0.45
HCAR3 P49019 2/20 0.45
PTGS2 P35354 2/20 0.44
ATM Q13315 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PTGS1 P23219 1/20 0.44
KDM4E B2RXH2 1/20 0.44
GLA P06280 1/20 0.44
LMNA P02545 1/20 0.44
RAF1 P04049 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7681987 1.00 MAPK1 (0.62) MAPK1VCAM1CES2CES1ALDH1A1
SCHEMBL3582037 0.90 SRD5A2 (0.55) MAPK1VCAM1CES2CES1ALDH1A1
SCHEMBL3582033 0.90 SRD5A2 (0.55) MAPK1VCAM1CES2CES1ALDH1A1
SCHEMBL7043142 0.84 CASP6 (0.64) PDK1CASP6HCAR3LMNA
SCHEMBL7043138 0.84 CASP6 (0.64) PDK1CASP6HCAR3LMNA
SCHEMBL8491427 0.83 VCAM1 (0.53) MAPK1VCAM1CES2CES1ALDH1A1
SCHEMBL8491434 0.83 MAPK1 (0.47) MAPK1VCAM1CES2CES1ALDH1A1
SCHEMBL5174175 0.82 MAPT (0.52) MAPK1CES2CES1ALDH1A1PDK1
SCHEMBL5174181 0.82 MAPT (0.52) MAPK1CES2CES1ALDH1A1PDK1
SCHEMBL11014183 0.81 MAPK1 (0.73) MAPK1VCAM1CES2CES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6469181-B1 PREPARING 2-OXINDOLES AND N-HYROXY-2- OXINDOLES VIA REDUCTION OF 2-NITROARYLMALONATE DIESTERS WITHOUT ISOLATION OF INTERMEDIATES CATALYTICA, INC. 2002-10-22 US disclosed
EP-0809631-A4 PROCESS FOR PREPARING 2-OXINDOLES AND N-HYDROXY-2-OXINDOLES CATALYTICA INC (US) 1998-07-08 EP disclosed
EP-0809631-A1 PROCESS FOR PREPARING 2-OXINDOLES AND N-HYDROXY-2-OXINDOLES CATALYTICA, INC. (US) 1997-12-03 EP disclosed
WO-1996023770-A1 PROCESS FOR PREPARING 2-OXINDOLES AND N-HYDROXY-2-OXINDOLES CATALYTICA, INC. (US) 1996-08-08 WO disclosed