SCHEMBL7682433

SCHEMBL7682433

Oc1cc(Cl)c(Cl)c(F)c1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 11/20 0.52
TSHR P16473 10/20 0.52
HPGD P15428 7/20 0.52
CYP3A4 P08684 7/20 0.52
HSP90AA1 P07900 2/20 0.52
ALDH1A1 P00352 4/20 0.44
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
CASP1 P29466 1/20 0.43
MAPK1 P28482 3/20 0.40
TDP1 Q9NUW8 1/20 0.39
ALOX15 P16050 3/20 0.34
ALOX12 P18054 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HIF1A Q16665 2/20 0.34
RECQL P46063 2/20 0.34
AKR1B1 P15121 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9115158 0.78 HSD17B10 (0.46) HSD17B10TSHRHPGDCYP3A4HSP90AA1
SCHEMBL11872648 0.75 CYP3A4 (0.50) HSD17B10TSHRHPGDCYP3A4HSP90AA1
SCHEMBL9643418 0.74 CYP3A4 (0.56) HSD17B10TSHRHPGDCYP3A4HSP90AA1
SCHEMBL25015441 0.73 HSD17B10 (0.41) HSD17B10TSHRHPGDCYP3A4HSP90AA1
SCHEMBL8761719 0.73 HSD17B10 (0.41) HSD17B10TSHRHPGDCYP3A4HSP90AA1
SCHEMBL1756490 0.72 CYP3A4 (0.40) HSD17B10TSHRHPGDCYP3A4HSP90AA1
SCHEMBL23409587 0.70 HSD17B10 (0.38) HSD17B10TSHRHPGDCYP3A4HSP90AA1
SCHEMBL29970962 0.70 HSD17B10 (0.38) HSD17B10TSHRHPGDCYP3A4HSP90AA1
SCHEMBL516276 0.70 CA9 (0.37) HSD17B10ALDH1A1MAPK1TDP1ALOX15
SCHEMBL202648 0.69 HSD17B10 (1.00) HSD17B10TSHRHPGDCYP3A4HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436961-B1 SUBSTANCE P RECEPTOR ANTAGONIST; 2-PHENYL-3-BENZYLAMINOPIPERIDINES PFIZER INC 2002-08-20 US disclosed
EP-0700384-A1 PROCESS FOR PREPARING AND RESOLVING 2-PHENYL-3-AMINOPIPERIDINE PFIZER (US) 1996-03-13 EP disclosed
WO-1994027966-A1 PROCESS FOR PREPARING AND RESOLVING 2-PHENYL-3-AMINOPIPERIDINE PFIZER INC. (US) 1994-12-08 WO disclosed
US-4020112-A WITH SULFUR TETRAFLUORIDE IN HYDROGEN FLUORIDE E. I. DU PONT DE NEMOURS AND COMPANY (US) 1977-04-26 US disclosed