SCHEMBL7683940

SCHEMBL7683940

Cc1cc(N(C)C)cc(C)c1Sc1nnn(CC(=O)C(CC(=O)OC(C)(C)C)NC(=O)SCc2ccccc2)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.35
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
IDO1 P14902 1/20 0.31
CNR2 P34972 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
BRD9 Q9H8M2 1/20 0.31
GHSR Q92847 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
ACE P12821 1/20 0.30
CASP1 P29466 1/20 0.30
CASP3 P42574 1/20 0.30
CASP7 P55210 1/20 0.30
CASP8 Q14790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8176683 0.90 TP53 (0.36) TP53MEN1KMT2ACASP1CASP3
Hydrochloric Acid SCHEMBL7689556 0.89 TP53 (0.36) TP53MEN1KMT2ACASP1CASP3
SCHEMBL7685546 0.82 CASP3 (0.38) TP53MEN1KMT2ACASP1CASP3
SCHEMBL7684199 0.82 TP53 (0.34) TP53MEN1KMT2ACASP1CASP3
SCHEMBL8165549 0.79 CASP1 (0.44) CASP1CASP3
Hydrochloric Acid SCHEMBL7695543 0.78 CASP3 (0.44) CASP1CASP3
SCHEMBL7686947 0.76 TP53 (0.37) TP53MEN1KMT2ACASP1CASP3
SCHEMBL8171557 0.76 ALDH1A1 (0.35) TP53KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL7680236 0.75 TP53 (0.33) TP53MEN1KMT2ACASP1CASP3
Hydrochloric Acid SCHEMBL8176793 0.75 UBE2M (0.35) TP53KMT2ACYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376484-B1 FOR PREVENTION AND/OR TREATMENT OF VARIOUS KINDS OF INFLAMMATORY DISEASE ONO PHARMACEUTICAL CO., LTD. (JP) 2002-04-23 US disclosed