SCHEMBL7684703

SCHEMBL7684703

COCc1ccc(Cl)c(C)c1NC(=O)c1ccc(C)nc1C(=O)NCC1CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 9/20 0.46
CNR2 P34972 5/20 0.46
PDE4B Q07343 2/20 0.36
PAK1 Q13153 2/20 0.36
PDE4A P27815 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
PTGES O14684 1/20 0.36
ACACB O00763 1/20 0.35
ACACA Q13085 1/20 0.35
P2RX7 Q99572 2/20 0.35
HTR3A P46098 1/20 0.35
HTR4 Q13639 1/20 0.35
KCNH2 Q12809 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7676296 0.88 PTGER4 (0.40) CNR1CNR2PDE4BPAK1PDE4A
SCHEMBL7677655 0.85 CNR2 (0.40) CNR1CNR2PDE4BPAK1PDE4A
SCHEMBL7677391 0.83 CNR1 (0.38) CNR1CNR2PDE4BPAK1PDE4A
SCHEMBL7675273 0.82 P2RX7 (0.39) CNR1CNR2PDE4BPAK1PDE4A
SCHEMBL678914 0.80 P2RX7 (0.38) CNR1CNR2PDE4BPAK1PDE4A
SCHEMBL7678800 0.78 ALDH1A1 (0.37) CNR1CNR2PDE4BPAK1PDE4A
SCHEMBL12808578 0.78 PAK1 (0.36) CNR1CNR2PDE4BPAK1PDE4A
SCHEMBL7675255 0.78 CNR1 (0.40) CNR1CNR2CYP3A4CYP2C9PTGES
SCHEMBL7679461 0.76 CNR1 (0.39) CNR1CNR2ACACBACACAMEN1
SCHEMBL7679296 0.75 CNR1 (0.38) CNR1CNR2CYP3A4CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472349-B1 Pyridine-2,3-dicarboxylic acid diamides BASF AKTIENGESELLSCHAFT (DE) 2002-10-29 US claimed