SCHEMBL7685246

SCHEMBL7685246

COc1ccc(Cl)cc1C1CC(=O)C=C(N)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.41
SRD5A1 P18405 2/20 0.39
PTGDR2 Q9Y5Y4 5/20 0.38
PTGDR Q13258 4/20 0.38
ADAM17 P78536 1/20 0.38
ALDH1A1 P00352 4/20 0.38
MAPT P10636 2/20 0.37
POLB P06746 2/20 0.37
TSHR P16473 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
CTSD P07339 1/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
GLA P06280 1/20 0.36
ALOX12 P18054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7685298 0.82 L3MBTL1 (0.45) TP53SRD5A1ALDH1A1MAPTPOLB
SCHEMBL34463208 0.80 MAP1LC3B (0.51) ALDH1A1RAB9AHTT
SCHEMBL7685135 0.79 TP53 (0.46) TP53PTGDR2PTGDRADAM17ALDH1A1
SCHEMBL14640344 0.70 PTGDR2 (0.62) PTGDR2PTGDRMAPTPOLBTSHR
SCHEMBL10257352 0.70 ALDH1A1 (0.44) TP53ADAM17ALDH1A1MAPTPOLB
SCHEMBL6804819 0.69 TP53 (0.57) TP53ALDH1A1MAPTPOLBTSHR
SCHEMBL24252872 0.68 PTGDR2 (0.46) TP53PTGDR2PTGDRADAM17ALDH1A1
SCHEMBL1093945 0.68 HTR2C (0.61) PTGDR2PTGDRHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL1266139 0.67 HTR2C (0.62) PTGDR2PTGDRHTR3EHTR3BHTR3A
SCHEMBL7680981 0.67 ALDH1A1 (0.33) ALDH1A1MAPTPOLBKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed