SCHEMBL7685490

SCHEMBL7685490

C=C(c1ccc(O)cc1)c1ccc(Br)cc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.75
GFER P55789 2/20 0.75
HTT P42858 2/20 0.75
HSD17B10 Q99714 2/20 0.75
GPR55 Q9Y2T6 1/20 0.75
ALOX15 P16050 2/20 0.65
ESR1 P03372 4/20 0.52
ESR2 Q92731 4/20 0.52
GLB1 P16278 1/20 0.50
CTRB1 P17538 1/20 0.50
CTRC Q99895 1/20 0.50
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
GAA P10253 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5049280 0.89 MAPT (0.55) MAPTGFERHTTHSD17B10GPR55
SCHEMBL6343638 0.89 MAPT (0.55) MAPTGFERHTTHSD17B10GPR55
SCHEMBL10942166 0.87 MAPT (1.00) MAPTGFERHTTHSD17B10GPR55
SCHEMBL824903 0.87 MAPT (1.00) MAPTGFERHTTHSD17B10GPR55
SCHEMBL17443 0.81
SCHEMBL6118114 0.81 ALOX15 (1.00) MAPTGFERHSD17B10ALOX15ESR1
SCHEMBL2287032 0.80 MEN1 (0.54) MAPTGFERHTTHSD17B10GPR55
SCHEMBL2279014 0.79 MAPT (0.58) MAPTGFERHTTHSD17B10GPR55
Formaldehyde SCHEMBL9616525 0.78 ALOX15 (0.81) MAPTGFERHTTHSD17B10GPR55
SCHEMBL10076323 0.78 MAPT (0.44) MAPTGFERHTTHSD17B10GPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed
CN-1158844-A Tertiary amines HOFFMANN LA ROCHE (CH) 1997-09-10 CN disclosed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed