SCHEMBL7686771

SCHEMBL7686771

CC(C)(C)S(=O)(=O)Nc1ccccc1.OBO

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.50
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
IL1RN P18510 1/20 0.44
ERAP1 Q9NZ08 1/20 0.44
NR3C2 P08235 2/20 0.43
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.41
PTPN11 Q06124 1/20 0.41
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5700054 0.92 KEAP1 (0.58) KEAP1CA1CA2IL1RNERAP1
SCHEMBL10116182 0.79 KMT2A (0.57) KMT2AMEN1ALDH1A1PKMMAPK1
SCHEMBL1358244 0.78 KEAP1 (0.83) KEAP1CA1CA2NR3C2ALDH1A1
SCHEMBL14571964 0.77 CA2 (0.54) KEAP1CA1CA2IL1RNERAP1
SCHEMBL13564999 0.76 CA1 (0.50) CA1CA2CA12CA9KMT2A
SCHEMBL19997241 0.76 CA2 (0.55) CA1CA2CA12CA9KMT2A
SCHEMBL27510736 0.74 NR3C2 (0.53) KEAP1CA1CA2IL1RNERAP1
SCHEMBL19997242 0.74 UQCRB (0.59) CA2KMT2AMEN1ALDH1A1PKM
SCHEMBL4599829 0.74 ALDH1A1 (0.58) KMT2AMEN1ALDH1A1SMN1; SMN2MAPT
SCHEMBL12601555 0.74 CA1 (0.57) CA1CA2CA12CA9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399627-B1 ANTICOAGULANTS; PROTHROMINASE, SERINE PROTEASE INHIBITOR; ACRYLAMIDE DERIVATIVES COR THERAPEUTICS, INC. 2002-06-04 US disclosed
EP-1159264-A2 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2001-12-05 EP disclosed
WO-2000047554-A2 INHIBITORS OF FACTOR Xa COR THERAPEUTICS INC. (US) 2000-08-17 WO disclosed