SCHEMBL7688580

SCHEMBL7688580

CCNc1cccnc1Nc1ccc2c(c1)CCN2c1nc2ccccc2[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.38
MAPT P10636 3/20 0.36
RAB9A P51151 1/20 0.36
CSNK1D P48730 1/20 0.36
CSNK1E P49674 1/20 0.36
PDE10A Q9Y233 1/20 0.36
FAAH O00519 1/20 0.35
PARP1 P09874 1/20 0.35
SYK P43405 2/20 0.35
ZAP70 P43403 1/20 0.35
KARS1 Q15046 1/20 0.35
EIF2AK3 Q9NZJ5 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
ERBB4 Q15303 1/20 0.34
HDAC11 Q96DB2 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
BACE1 P56817 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL569493 0.73 ROCK1 (0.47) MAPTRAB9AHDAC11HDAC6MEN1
SCHEMBL570508 0.71 MAPT (0.36) MAPTRAB9APDE10ASMN1; SMN2MEN1
SCHEMBL1701449 0.71 PDE10A (0.37) MAPTRAB9APDE10AFAAHSMN1; SMN2
SCHEMBL7694281 0.70 SYK (0.42) SYKEIF2AK3EGFRERBB2ERBB4
SCHEMBL7689084 0.70 GRM5 (0.45) GRM5SMN1; SMN2
SCHEMBL1018884 0.70 ALDH1A1 (0.53) MAPTRAB9APDE10ASMN1; SMN2HDAC11
SCHEMBL12473779 0.67 ACSS2 (0.39) MAPTRAB9ASMN1; SMN2HDAC11HDAC6
SCHEMBL14889094 0.67 ACHE (0.36) MAPTRAB9ASMN1; SMN2HDAC11HDAC6
SCHEMBL7702320 0.66 GRM5 (0.41) GRM5MAPTRAB9APDE10ASMN1; SMN2
SCHEMBL7688852 0.63 GRM5 (0.55) GRM5MAPTRAB9ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed