SCHEMBL7688612

SCHEMBL7688612

O=C(O)c1cc(F)c2cccnc2c1O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.60
L3MBTL1 Q9Y468 8/20 0.57
ALDH1A1 P00352 5/20 0.57
MEN1 O00255 5/20 0.57
KMT2A Q03164 5/20 0.57
TDP1 Q9NUW8 4/20 0.57
LMNA P02545 3/20 0.57
MAPT P10636 3/20 0.57
IDO1 P14902 2/20 0.57
TDO2 P48775 2/20 0.57
POLB P06746 1/20 0.57
THRB P10828 1/20 0.57
PKM P14618 1/20 0.57
RECQL P46063 1/20 0.57
BLM P54132 1/20 0.57
CASP6 P55212 1/20 0.57
KDM4A O75164 2/20 0.54
EGLN1 Q9GZT9 2/20 0.54
KDM6B O15054 1/20 0.54
KDM6A O15550 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2015831 0.86 L3MBTL1 (0.60) KDM4EL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL28463407 0.85 KDM4E (0.74) KDM4EL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL4061248 0.81 KDM4E (0.66) KDM4EL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL2143785 0.81 KDM4E (0.78) KDM4EL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL16207365 0.80 KDM4E (0.62) KDM4EL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL5306342 0.79 KDM4E (0.59) KDM4EL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL8883998 0.78 ENPP2 (0.60) KDM4EL3MBTL1ALDH1A1KDM4AEGLN1
SCHEMBL8882706 0.77 ENPP2 (0.58) KDM4EL3MBTL1ALDH1A1KDM4AEGLN1
SCHEMBL8882696 0.77 ENPP2 (0.58) KDM4EL3MBTL1ALDH1A1KDM4AEGLN1
SCHEMBL485003 0.76 HSD17B10 (0.67) KDM4EALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6500842-B1 N-((4-CHLOROPHENYL)METHYL)-8-HYDROXY-7-QUINOLINECARBOXAMIDE ADMINISTERED AS VIRICIDES AGAINST HERPES VIRUS PHARMACIA & UPJOHN COMPANY 2002-12-31 US disclosed
US-6310211-B1 ANTI-VIRAL ACTIVITY AGAINST HERPES VIRUS, CYTOMEGALOVIRUS. MANY OF THESE COMPOUNDS ARE ALSO ACTIVE AGAINST VARICELLA ZOSTER VIRUS, EPSTEIN-BARR VIRUS, HERPES SIMPLEX VIRUS AND HUMAN HERPES VIRUS TYPE 8 PHARMACIA & UPJOHN COMPANY 2001-10-30 US disclosed
US-6252080-B1 HERPES, CYTOMEGALO VIRUS PHARMACIA & UPJOHN COMPANY 2001-06-26 US disclosed
US-6211376-B1 HERPES VIRUS, CYTOMEGALO VIRUS, VARICELLA-ZOSTER VIRUS,EPSTEIN-BARR VIRUS PHARMACIA & UPJOHN COMPANY 2001-04-03 US disclosed
EP-0927164-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1999-07-07 EP disclosed
WO-1998011073-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1998-03-19 WO disclosed