SCHEMBL7689388

SCHEMBL7689388

Cc1n[nH]c2c1C(=O)CC(c1cc(Cl)sc1Cl)C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.34
ALDH1A1 P00352 2/20 0.34
ALPL P05186 1/20 0.34
MAPK1 P28482 1/20 0.34
PIM1 P11309 4/20 0.33
CLK4 Q9HAZ1 4/20 0.33
ERBB2 P04626 1/20 0.33
FLT3 P36888 1/20 0.33
MAP4K2 Q12851 1/20 0.33
AXL P30530 1/20 0.32
PTK2B Q14289 1/20 0.32
MAPKAPK5 Q8IW41 1/20 0.32
SRPK1 Q96SB4 1/20 0.32
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CSNK1G1 Q9HCP0 1/20 0.31
RXFP1 Q9HBX9 1/20 0.30
USP2 O75604 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7689368 0.79 PIM1 (0.45) TP53ALDH1A1MAPK1PIM1CLK4
SCHEMBL7683237 0.78 SMN1; SMN2 (0.48) TP53ALDH1A1MAPK1PIM1CLK4
Hydrochloric Acid SCHEMBL7687660 0.78 PIM1 (0.44) TP53ALDH1A1MAPK1PIM1CLK4
SCHEMBL6804202 0.75 LMNA (0.30) HSD17B10LMNA
SCHEMBL7689241 0.75 HCAR2 (0.48) TP53ALDH1A1ALPLALOX15TSHR
Hydrochloric Acid SCHEMBL7689302 0.74 LMNA (0.30) HSD17B10LMNA
Hydrochloric Acid SCHEMBL7689305 0.74 LMNA (0.30) HSD17B10LMNA
SCHEMBL7683192 0.73 ALDH1A1 (0.33) TP53ALDH1A1ALPLMAPK1PIM1
SCHEMBL7682852 0.73 HSD17B10 (0.39) TP53ALDH1A1ALPLALOX15TSHR
SCHEMBL7678938 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed