SCHEMBL7690365

SCHEMBL7690365

CCOC(=O)C1=C(C)NC(=S)NC1c1ccc(OC)c(O)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GUSB P08236 1/20 0.74
DHFR P00374 2/20 0.64
CA1 P00915 4/20 0.63
CA2 P00918 4/20 0.63
CA12 O43570 1/20 0.63
CA7 P43166 1/20 0.63
CA9 Q16790 1/20 0.63
GAA P10253 3/20 0.61
ALDH1A1 P00352 5/20 0.59
ADORA2B P29275 3/20 0.59
POLB P06746 1/20 0.59
MAPT P10636 2/20 0.59
MAPK1 P28482 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
TSHR P16473 3/20 0.57
RAB9A P51151 1/20 0.57
ALOX12 P18054 1/20 0.56
HTT P42858 1/20 0.56
ALOX15 P16050 1/20 0.55
CASP1 P29466 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13419868 0.91 GAA (0.70) GUSBDHFRCA1CA2CA12
SCHEMBL4669190 0.91 ALDH1A1 (0.67) GUSBDHFRCA1CA2CA12
SCHEMBL26671671 0.84 ALDH1A1 (0.64) GUSBDHFRCA1CA2CA12
SCHEMBL3168404 0.82 CA1 (0.79) GUSBDHFRCA1CA2CA12
SCHEMBL10279642 0.82 DHFR (0.74) GUSBDHFRCA1CA2CA12
SCHEMBL5380810 0.82 DHFR (0.79) GUSBDHFRCA1CA2CA12
SCHEMBL26671696 0.81 ALDH1A1 (0.60) GUSBDHFRCA1CA2CA12
SCHEMBL29793923 0.81 ALDH1A1 (0.60) GUSBDHFRCA1CA2CA12
SCHEMBL10112977 0.81 DHFR (0.72) DHFRCA1CA2CA12CA7
SCHEMBL28558189 0.81 DHFR (0.81) DHFRCA1CA2CA12CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002066443-A2 2-THIOXO-1,2,3,4-TETRAHYDROPYRIMIDINE DERIVATIVES ONO PHARMACEUTICAL CO., LTD. (JP) 2002-08-29 WO disclosed