SCHEMBL7696758

SCHEMBL7696758

CC(C)(C)c1cc(Nc2nc3cc4ccccc4cc3nc2NCC2CCN(Cc3ccccc3)CC2)n(-c2cccc(F)c2)n1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.40
NTRK1 P04629 1/20 0.39
ACHE P22303 7/20 0.39
BACE1 P56817 3/20 0.38
MAPK14 Q16539 2/20 0.38
KDM1A O60341 1/20 0.38
EHMT2 Q96KQ7 1/20 0.38
RCOR1 Q9UKL0 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 1/20 0.38
CHRM4 P08173 1/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
PIM1 P11309 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7700675 0.81 MAPK14 (0.43) NTRK1MAPK14
SCHEMBL7690441 0.78 MAPK14 (0.47) NTRK1MAPK14
SCHEMBL7691048 0.78 MAPK14 (0.42) MAPK14MEN1KMT2A
SCHEMBL7691122 0.77 MAPK14 (0.50) MAPK14
SCHEMBL7697564 0.77 MAPK14 (0.41) NTRK1MAPK14
SCHEMBL7693923 0.77 MAPK14 (0.45) NTRK1MAPK14
SCHEMBL7694525 0.76 MAPK14 (0.39) NTRK1MAPK14
SCHEMBL7697861 0.76 MAPK14 (0.47) NTRK1MAPK14
SCHEMBL7696568 0.76 MAPK14 (0.41) NTRK1MAPK14
SCHEMBL7694572 0.74 MAPT (0.39) TP53NTRK1MAPK14MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002094796-A2 BENZO[G]QUINOXALINE DERIVATIVES AS EFFECTIVE COMPOUNDS AGAINST INFECTIOUS DISEASES AXXIMA PHARMACEUTICALS AG (DE) 2002-11-28 WO disclosed