SCHEMBL7696975

SCHEMBL7696975

CCc1cccc2c(C3CCN(CCC4CCN(/C=C/C(=O)c5ccc(Cl)c(Cl)c5)CC4)CC3)c[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.49
CCR2 P41597 15/20 0.47
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
OPRL1 P41146 1/20 0.41
DRD2 P14416 3/20 0.38
HTR2A P28223 3/20 0.38
DRD3 P35462 3/20 0.38
KCNH2 Q12809 1/20 0.38
CACNA1I Q9P0X4 1/20 0.38
HTR1A P08908 1/20 0.37
HTR1B P28222 1/20 0.37
HTR2C P28335 1/20 0.37
HTR1E P28566 1/20 0.37
HTR1F P30939 1/20 0.37
HTR7 P34969 1/20 0.37
HTR2B P41595 1/20 0.37
HTR6 P50406 1/20 0.37
CCR5 P51681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702484 0.93 OPRM1 (0.49) SLC2A1CCR2OPRM1OPRK1OPRL1
SCHEMBL7701223 0.92 CCR2 (0.49) SLC2A1CCR2OPRM1OPRK1OPRL1
SCHEMBL7705374 0.85 SLC2A1 (0.46) SLC2A1CCR2DRD2HTR2ADRD3
SCHEMBL7700232 0.83 SLC2A1 (0.69) SLC2A1CCR2
SCHEMBL7702546 0.83 SLC2A1 (0.52) SLC2A1CCR2DRD2HTR2ADRD3
SCHEMBL7700045 0.82 CCR2 (0.56) SLC2A1CCR2DRD2HTR2ADRD3
SCHEMBL7694620 0.82 CCR2 (0.56) SLC2A1CCR2DRD2HTR2ADRD3
SCHEMBL7701921 0.82 CCR2 (0.56) SLC2A1CCR2DRD2HTR2ADRD3
SCHEMBL7699820 0.81 CCR2 (0.58) SLC2A1CCR2DRD2HTR2AHTR1A
SCHEMBL7702544 0.80 CCR2 (0.62) SLC2A1CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002079190-A1 3-SUBSTITUTED INDOLES AS CHEMOKINE ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-10-10 WO disclosed