SCHEMBL7697015

SCHEMBL7697015

CS(=O)(=O)N(CC12CN(CCc3ccccc3)CCC1CN(Cc1ccccc1)C2)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 1/20 0.42
OPRM1 P35372 8/20 0.41
OPRD1 P41143 7/20 0.41
OPRK1 P41145 6/20 0.41
ADRA1A P35348 3/20 0.41
ADRA1B P35368 3/20 0.41
CHRM3 P20309 2/20 0.40
SLC22A1 O15245 1/20 0.40
NR1I2 O75469 1/20 0.40
ABCB1 P08183 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD2 P14416 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
MAOA P21397 1/20 0.40
DRD4 P21917 1/20 0.40
MAOB P27338 1/20 0.40
HRH1 P35367 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7700744 0.89 KCNH2 (0.40) KCNH2HTR2AHTR2COPRM1SIGMAR1
SCHEMBL7695892 0.81 HTR2A (0.45) KCNH2HTR2AHTR2CDRD2ACHE
SCHEMBL7695908 0.79 HTR2A (0.43) KCNH2HTR2AHTR2COPRM1ADRA1A
SCHEMBL7701553 0.79 OPRM1 (0.41) KCNH2HTR2AHTR2COPRM1OPRD1
SCHEMBL7694829 0.78 HTR2A (0.46) KCNH2HTR2AHTR2CSIGMAR1ACHE
SCHEMBL7707462 0.76 ACHE (0.44) KCNH2HTR2AHTR2CACHE
SCHEMBL7700571 0.74 ACHE (0.42) KCNH2HTR2AHTR2CDRD2SIGMAR1
SCHEMBL7701119 0.72 OPRM1 (0.56) KCNH2OPRM1OPRD1OPRK1ADRA1A
SCHEMBL7698615 0.72 LTA4H (0.48) HTR2AMAOADRD4MAOBSIGMAR1
SCHEMBL7697370 0.72 OPRM1 (0.56) KCNH2OPRM1OPRD1OPRK1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002046187-A1 ANALGESIC DIAZABICYCLO[4.3.0]NONANES SEPRACOR, INC. (US) 2002-06-13 WO disclosed