SCHEMBL7698333

SCHEMBL7698333

CC[Si](CC)(CC)c1[nH]c2ccc(C(F)(F)F)cc2c1CCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
MAPT P10636 3/20 0.43
NPSR1 Q6W5P4 3/20 0.43
KIF11 P52732 1/20 0.42
MDH2 P40926 1/20 0.42
CCNB2 O95067 2/20 0.41
CDK1 P06493 2/20 0.41
CCNB1 P14635 2/20 0.41
GSK3B P49841 2/20 0.41
CDK5 Q00535 2/20 0.41
CDK5R1 Q15078 2/20 0.41
CCNB3 Q8WWL7 2/20 0.41
GAA P10253 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
DDR1 Q08345 3/20 0.39
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL891994 0.77 KIF11 (0.46) MEN1KMT2AMAPTKIF11KDM4E
SCHEMBL7679735 0.77 KIF11 (0.46) MEN1KMT2AKIF11KDM4E
SCHEMBL892668 0.77 CYP2C9 (0.47) ALDH1A1MEN1KMT2AKIF11KDM4E
SCHEMBL30532272 0.77 CYP2C9 (0.47) ALDH1A1MEN1KMT2AKIF11KDM4E
SCHEMBL25366837 0.74 CCNB2 (0.43) ALDH1A1MEN1KMT2AMAPTNPSR1
SCHEMBL30642000 0.74 CCNB2 (0.43) ALDH1A1MEN1KMT2AMAPTNPSR1
SCHEMBL15313180 0.73 KIF11 (0.43) MEN1KMT2AKIF11DDR1KDM4E
SCHEMBL14074159 0.68 MAPT (0.57) ALDH1A1MEN1KMT2AMAPTNPSR1
SCHEMBL8665875 0.68 MAPT (0.51) ALDH1A1MEN1KMT2AMAPTNPSR1
SCHEMBL7957008 0.67 ADRA1D (0.62) ALDH1A1KMT2AMAPTNPSR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350757-B1 Beta-carboline compounds LES LABORATOIRES SERVIER (FR) 2002-02-26 US disclosed
EP-1070716-A1 Beta-carboline derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2001-01-24 EP disclosed