SCHEMBL7679735

SCHEMBL7679735

CC[Si](CC)(CC)c1[nH]c2ccc(C(F)(F)F)cc2c1CCN

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
HTR1D P28221 3/20 0.41
HTR6 P50406 2/20 0.41
CHUK O15111 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTR7 P34969 1/20 0.41
HTR3A P46098 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
HRH1 P35367 1/20 0.38
HRH4 Q9H3N8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL891994 0.87 KIF11 (0.46) KIF11MEN1KMT2AHTR6CHUK
SCHEMBL30532272 0.87 CYP2C9 (0.47) KIF11MEN1KMT2ACHUKCYP1A2
SCHEMBL892668 0.87 CYP2C9 (0.47) KIF11MEN1KMT2ACHUKCYP1A2
SCHEMBL15313180 0.82 KIF11 (0.43) KIF11MEN1KMT2AHTR6CHUK
SCHEMBL7698333 0.77 ALDH1A1 (0.43) KIF11MEN1KMT2AKDM4E
SCHEMBL14499883 0.72 GHSR (0.43) KIF11MEN1KMT2ACHUKHSD17B10
SCHEMBL22417826 0.71 MEN1 (0.54) KIF11MEN1KMT2AHTR6CHUK
SCHEMBL4951539 0.70 HTT (0.40) KIF11MEN1KMT2ACHUKHSD17B10
SCHEMBL18932887 0.69 ALDH1A1 (0.44) KIF11MEN1KMT2AHSD17B10KDM4E
SCHEMBL412032 0.67 KIF11 (0.81) KIF11MEN1KMT2ACHUKKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350757-B1 Beta-carboline compounds LES LABORATOIRES SERVIER (FR) 2002-02-26 US disclosed
EP-1070716-A1 Beta-carboline derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2001-01-24 EP disclosed