SCHEMBL7698337

SCHEMBL7698337

Cc1ccccc1OCCN(C)CCc1ccc(N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.51
SIGMAR1 Q99720 2/20 0.45
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
ALDH1A1 P00352 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CYBB P04839 1/20 0.42
NCF1 P14598 1/20 0.42
HTR1D P28221 2/20 0.42
HTR1B P28222 2/20 0.42
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.40
CACNA1F O60840 1/20 0.40
CHRM2 P08172 1/20 0.40
ACHE P22303 1/20 0.40
AGTR1 P30556 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7697582 0.84 KCNH2 (0.52) KCNH2SIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL13459968 0.84 NPC1 (0.54) ALDH1A1DRD2DRD4GAA
SCHEMBL23074694 0.83 HTR1B (0.54) ALDH1A1NPSR1CYBBNCF1HTR1D
SCHEMBL7702574 0.81 KCNH2 (0.69) KCNH2SIGMAR1ALDH1A1
SCHEMBL10726453 0.81 LMNA (0.50) KCNH2SIGMAR1SLC6A3ALDH1A1CHRM2
Hydrochloric Acid SCHEMBL7705362 0.80 KCNH2 (0.67) KCNH2SIGMAR1ALDH1A1
SCHEMBL7024969 0.79 KCNH2 (0.73) KCNH2SIGMAR1CACNA1FCHRM2ACHE
SCHEMBL7695482 0.79 KCNH2 (0.70) KCNH2ALDH1A1CACNA1FCHRM2ACHE
Hydrochloric Acid SCHEMBL7696220 0.78 KCNH2 (0.69) KCNH2ALDH1A1CACNA1FCHRM2ACHE
SCHEMBL7700695 0.77 SIGMAR1 (0.44) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037871-B1 NOVEL ANTIARRHYTHMIC COMPOUNDS GYOGYSZERKUTATO INTEZET (HU) 2002-07-03 EP disclosed
US-6265445-B1 CARDIOVASCULAR DISORDERS GYOGYSZERKUTATO INTEZET KFT (HU) 2001-07-24 US disclosed
EP-1037871-A1 NOVEL ANTIARRHYTHMIC COMPOUNDS GYOGYSZERKUTATO INTEZET KFT. (HU) 2000-09-27 EP disclosed
WO-1999029655-A1 NOVEL ANTIARRHYTHMIC COMPOUNDS Gyógyszerkutató Intézet Kft. (HU) 1999-06-17 WO disclosed