SCHEMBL7700599

SCHEMBL7700599

O=C(O)Nc1cc(N2CC=CC2)c(I)cc1[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
MAPT P10636 10/20 0.38
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
GAA P10253 2/20 0.37
WDR5 P61964 1/20 0.37
ALDH1A1 P00352 8/20 0.36
POLB P06746 2/20 0.36
MAPK1 P28482 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
GLA P06280 1/20 0.36
CASP3 P42574 1/20 0.36
HTT P42858 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
KMT2A Q03164 2/20 0.36
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7704017 0.86 WDR5 (0.49) SMN1; SMN2MAPTLMNAGAAWDR5
SCHEMBL7148612 0.82 MAPK1 (0.37) SMN1; SMN2MAPTLMNAGAAWDR5
SCHEMBL7702872 0.79 MAPT (0.43) SMN1; SMN2MAPTLMNATP53ALDH1A1
SCHEMBL7698657 0.76 MAPT (0.49) HCAR3SMN1; SMN2MAPTLMNATP53
SCHEMBL7703607 0.76 MAPT (0.40) SMN1; SMN2MAPTTP53ALDH1A1MAPK1
SCHEMBL6608481 0.75 CXCR2 (0.43) HCAR3MAPTLMNAGAAALDH1A1
SCHEMBL6611671 0.74 MAPT (0.59) SMN1; SMN2MAPTLMNAALDH1A1POLB
SCHEMBL6609390 0.73 MAPT (0.60) SMN1; SMN2MAPTLMNAGAAALDH1A1
SCHEMBL7143246 0.72 ALDH1A1 (0.45) SMN1; SMN2MAPTLMNAGAAWDR5
SCHEMBL27485058 0.72 SMN1; SMN2 (0.35) SMN1; SMN2MAPTLMNAGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed