SCHEMBL7700988

SCHEMBL7700988

CCOC(=O)c1cc(CN2CCOCC2)nn1C

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
TSHR P16473 4/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MAPK1 P28482 1/20 0.45
STAT3 P40763 1/20 0.45
RAB9A P51151 1/20 0.45
KDM4E B2RXH2 1/20 0.44
POLB P06746 2/20 0.44
PIK3CA P42336 1/20 0.44
HSD17B10 Q99714 1/20 0.43
TP53 P04637 1/20 0.43
CASP7 P55210 1/20 0.42
CASP6 P55212 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2210279 0.83 HTT (0.43) ALDH1A1LMNAMAPTSMN1; SMN2KDM4E
SCHEMBL15651814 0.82 CXCR4 (0.42) LMNASMN1; SMN2KDM4E
SCHEMBL19635510 0.80 POLB (0.47) ALDH1A1LMNASMN1; SMN2RAB9AKDM4E
SCHEMBL973113 0.78 LMNA (0.50) ALDH1A1LMNAMAPTSMN1; SMN2MAPK1
SCHEMBL7699075 0.77 LMNA (0.49) ALDH1A1LMNAMAPTSMN1; SMN2MAPK1
SCHEMBL19635528 0.76 POLB (0.47) ALDH1A1LMNASMN1; SMN2KDM4EPOLB
SCHEMBL859 0.76 POLB (0.50) ALDH1A1LMNAMAPTSMN1; SMN2MAPK1
SCHEMBL5900613 0.76 LMNA (0.48) ALDH1A1LMNAMAPTSMN1; SMN2MAPK1
SCHEMBL1810598 0.75 ALDH1A1 (0.47) ALDH1A1TSHRLMNAMAPTSMN1; SMN2
SCHEMBL7703155 0.74 LMNA (0.47) LMNAMAPTSMN1; SMN2RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2530078-A1 THIAZOLE DERIVATIVE Takeda Pharmaceutical Company Limited (JP) 2012-12-05 EP disclosed
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed