SCHEMBL7701314

SCHEMBL7701314

Cc1[nH]c2ccccc2c1C1CCN(CCC2CCN(/C=C/C(=O)c3ccc(Cl)c(Cl)c3)CC2)CC1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.46
KCNH2 Q12809 3/20 0.46
HDAC1 Q13547 2/20 0.46
SLC2A1 P11166 1/20 0.44
OPRM1 P35372 2/20 0.41
OPRK1 P41145 2/20 0.41
OPRD1 P41143 1/20 0.40
OPRL1 P41146 1/20 0.40
ACHE P22303 2/20 0.40
BCHE P06276 1/20 0.40
CACNA1I Q9P0X4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7701149 0.93 OPRM1 (0.49) CCR2KCNH2HDAC1OPRM1OPRK1
SCHEMBL7702984 0.90 CCR2 (0.40) CCR2KCNH2HDAC1SLC2A1OPRM1
SCHEMBL7701223 0.80 CCR2 (0.49) CCR2KCNH2SLC2A1OPRM1OPRK1
SCHEMBL7700232 0.80 SLC2A1 (0.69) CCR2SLC2A1
SCHEMBL7702546 0.79 SLC2A1 (0.52) CCR2SLC2A1
SCHEMBL7701921 0.78 CCR2 (0.56) CCR2SLC2A1
SCHEMBL7696975 0.78 SLC2A1 (0.49) CCR2KCNH2SLC2A1OPRM1OPRK1
SCHEMBL7700045 0.76 CCR2 (0.56) CCR2SLC2A1
SCHEMBL7694620 0.76 CCR2 (0.56) CCR2SLC2A1
SCHEMBL7705374 0.76 SLC2A1 (0.46) CCR2KCNH2SLC2A1CACNA1I

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002079190-A1 3-SUBSTITUTED INDOLES AS CHEMOKINE ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-10-10 WO disclosed