SCHEMBL7701331

SCHEMBL7701331

Nc1cc(C#Cc2ccccc2)c(OCC2COC(=O)O2)cc1NC(=O)O

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.34
ALDH1A1 P00352 1/20 0.33
GRM5 P41594 4/20 0.33
FFAR1 O14842 5/20 0.32
VCP P55072 2/20 0.31
PKM P14618 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7140004 0.89 RORC (0.32) PTGDR2ALDH1A1GRM5FFAR1
SCHEMBL7145378 0.76 ADRA2A (0.35) ALDH1A1
SCHEMBL7704027 0.76 FFAR1 (0.49) PTGDR2ALDH1A1FFAR1GAA
SCHEMBL7143235 0.73 MAPK14 (0.39)
SCHEMBL7143481 0.72 RORC (0.35) GRM5
SCHEMBL1324044 0.67 TDP1 (0.61) ALDH1A1FFAR1PKMGAA
SCHEMBL7146584 0.67
SCHEMBL7699272 0.66 GAA (0.39) ALDH1A1GRM5FFAR1GAA
SCHEMBL9999540 0.66 ALDH1A1 (0.64) ALDH1A1PKM
SCHEMBL7703655 0.65 PIK3CA (0.38) ALDH1A1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed