SCHEMBL7704027

SCHEMBL7704027

N#CCOc1cc(NC(=O)O)c(N)cc1C#Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 4/20 0.49
PTGDR2 Q9Y5Y4 5/20 0.40
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 2/20 0.35
CYP2C9 P11712 2/20 0.35
MEN1 O00255 2/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 2/20 0.35
KMT2A Q03164 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
LMNA P02545 2/20 0.35
RAB9A P51151 1/20 0.35
BRPF1 P55201 1/20 0.34
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7138333 0.87 FFAR1 (0.44) FFAR1PTGDR2
SCHEMBL7698583 0.83 FFAR1 (0.43) FFAR1PTGDR2NPC1CYP2C9MEN1
SCHEMBL15459105 0.78 FFAR1 (0.52) FFAR1PTGDR2KDM4EALDH1A1NPC1
SCHEMBL7704399 0.78 FFAR1 (0.40) FFAR1PTGDR2MEN1KMT2ALMNA
SCHEMBL7701331 0.76 PTGDR2 (0.34) FFAR1PTGDR2ALDH1A1GAA
SCHEMBL7699272 0.74 GAA (0.39) FFAR1KDM4EALDH1A1NPC1CYP2C9
SCHEMBL29608299 0.73 FFAR1 (0.67) FFAR1PTGDR2KDM4EALDH1A1NPC1
SCHEMBL7141263 0.72 PTGDR2 (0.41) FFAR1PTGDR2CYP2C9MAPTHPGD
SCHEMBL7142632 0.72 VCP (0.39) PTGDR2KDM4EHPGDHTT
SCHEMBL7142218 0.72 VCP (0.40) PTGDR2KDM4EHPGDKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed