SCHEMBL7701725

SCHEMBL7701725

Cc1ncc2cn[nH]c(=O)n12

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.33
DYRK1A Q13627 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
TBXAS1 P24557 1/20 0.31
XDH P47989 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11315951 0.77 TDP1 (0.33) ALDH1A1
SCHEMBL25408012 0.73 MAPK8 (0.33) MAPK8DYRK1ACLK4DYRK1BXDH
SCHEMBL11029949 0.72 SMN1; SMN2 (0.33) MAPK8DYRK1ACLK4DYRK1BTBXAS1
SCHEMBL7702569 0.68 XDH (0.33) XDHALDH1A1
SCHEMBL11306298 0.67 PDE5A (0.49) ALDH1A1
SCHEMBL21434271 0.64 GSK3A (0.36) ALDH1A1
SCHEMBL25410369 0.64 CHEK1 (0.37) XDHALDH1A1
SCHEMBL31687853 0.63 CHEK1 (0.32)
SCHEMBL31136330 0.61 TNKS (0.33) ALDH1A1
SCHEMBL7704795 0.60 ALDH1A1 (0.32) XDHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002081473-A1 SUBSTITUTED AZOLOAZIN(THI)ONES BAYER CROPSCIENCE AG (DE) 2002-10-17 WO disclosed
US-RE30511-E ENZYME INHIBITOR, HERBICIDE, CYCLIZATION AMERICAN CYANAMID COMPANY (US) 1981-02-10 US disclosed
US-4168964-A HERBICIDES AMERICAN CYANAMID COMPANY (US) 1979-09-25 US disclosed
US-4124766-A INTERMEDIATES FOR PHOSPHODIESTERASE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1978-11-07 US disclosed
US-4107307-A ENZYME INHIBITORS, HERBICIDES, RING CLOSURE AMERICAN CYANAMID COMPANY (US) 1978-08-15 US disclosed