SCHEMBL7702569

SCHEMBL7702569

Cc1nc(C)n2c(=O)[nH]ncc12

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PDE5A O76074 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE1C Q14123 1/20 0.33
PDE3A Q14432 1/20 0.33
TSHR P16473 1/20 0.32
CHEK1 O14757 2/20 0.31
ADORA1 P30542 1/20 0.31
POLB P06746 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
PARP10 Q53GL7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11307782 0.80 XDH (0.31) XDHPDE5APDE1APDE1BPDE3B
SCHEMBL7702068 0.78 KDM4E (0.35) ALDH1A1PARP10
SCHEMBL11304872 0.77 PDE1A (0.46) XDHALDH1A1PDE5APDE1APDE1B
SCHEMBL11080771 0.77 PDE10A (0.43) XDHPDE5APDE1APDE1BPDE3B
SCHEMBL11563762 0.75 KMT2A (0.40) PDE5APDE1APDE1BPDE3BPDE1C
SCHEMBL11560504 0.74 NOTUM (0.43) XDHPDE5APDE1APDE1BPDE3B
SCHEMBL11304795 0.71 APOBEC3G (0.44) XDHALDH1A1POLB
SCHEMBL25410369 0.70 CHEK1 (0.37) XDHALDH1A1TSHRCHEK1PARP10
SCHEMBL31687853 0.69 CHEK1 (0.32) CHEK1
SCHEMBL7701725 0.68 MAPK8 (0.33) XDHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002081473-A1 SUBSTITUTED AZOLOAZIN(THI)ONES BAYER CROPSCIENCE AG (DE) 2002-10-17 WO disclosed
US-RE30511-E ENZYME INHIBITOR, HERBICIDE, CYCLIZATION AMERICAN CYANAMID COMPANY (US) 1981-02-10 US disclosed
US-4168964-A HERBICIDES AMERICAN CYANAMID COMPANY (US) 1979-09-25 US disclosed
US-4124766-A INTERMEDIATES FOR PHOSPHODIESTERASE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1978-11-07 US disclosed
US-4107307-A ENZYME INHIBITORS, HERBICIDES, RING CLOSURE AMERICAN CYANAMID COMPANY (US) 1978-08-15 US disclosed