SCHEMBL7702344

SCHEMBL7702344

Clc1ccc(C2=NCCc3ccccc32)cn1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.47
NOS3 P29474 1/20 0.44
NOS2 P35228 1/20 0.44
MAPK10 P53779 11/20 0.43
MAPK9 P45984 2/20 0.39
MAPK14 Q16539 2/20 0.39
MAPK8 P45983 1/20 0.39
CYP2A6 P11509 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
PIK3CD O00329 1/20 0.38
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702043 0.82 NOS3 (0.44) MAOANOS3NOS2MAPK10MAPK9
SCHEMBL28542282 0.81 MAPK10 (0.50) MAOANOS3NOS2MAPK10MAPK9
SCHEMBL7705693 0.81 NOS3 (0.42) MAOANOS3NOS2MAPK10MAPK9
SCHEMBL7697815 0.78 NOS3 (0.41) MAOANOS3NOS2MAPK10MAPK9
SCHEMBL7698312 0.77 NOS3 (0.43) MAOANOS3NOS2CA1CA2
SCHEMBL163051 0.77 MAPK10 (0.55) MAOANOS3NOS2MAPK10MAPK9
SCHEMBL29384557 0.77 MAPK10 (0.55) MAOANOS3NOS2MAPK10MAPK9
SCHEMBL28190730 0.77 NOS3 (0.55) MAOANOS3NOS2MAPK10MAPK9
SCHEMBL10425795 0.75 MAPK10 (0.69) MAPK10MAPK9MAPK14MAPK8CA1
Hydrochloric Acid SCHEMBL27495714 0.75 MAPK10 (0.54) MAOANOS3NOS2MAPK10MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed