SCHEMBL7705693

SCHEMBL7705693

CN(C)c1ccc(C2=NCCc3ccccc32)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.42
NOS2 P35228 1/20 0.42
MAPK10 P53779 6/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.38
MAP3K11 Q16584 1/20 0.38
APP P05067 2/20 0.38
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
TDO2 P48775 1/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK14 Q16539 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702043 0.84 NOS3 (0.44) NOS3NOS2MAPK10MAOANPC1
SCHEMBL7702407 0.83 TACR1 (0.40) NOS3NOS2MAPK10MAOAPOLB
SCHEMBL7702344 0.81 MAOA (0.47) NOS3NOS2MAPK10MAOANPC1
SCHEMBL7697815 0.80 NOS3 (0.41) NOS3NOS2MAPK10MAOAALDH1A1
SCHEMBL13805616 0.76 NOS3 (0.49) NOS3NOS2MAPK10MAOANPC1
SCHEMBL7698312 0.76 NOS3 (0.43) NOS3NOS2MAOAALDH1A1LMNA
SCHEMBL7704878 0.76 CNR2 (0.47) TDO2
SCHEMBL29384557 0.76 MAPK10 (0.55) NOS3NOS2MAPK10MAOAALDH1A1
SCHEMBL163051 0.76 MAPK10 (0.55) NOS3NOS2MAPK10MAOAALDH1A1
Hydrochloric Acid SCHEMBL27495714 0.74 MAPK10 (0.54) NOS3NOS2MAPK10MAOAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1098260-C 2,4-diaminopyrimidine derivatives BASLIR PHARMACEUTICALS AG (CH) 2003-01-08 CN disclosed
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
CN-1218465-A 2,4-diaminopyrimidine derivatives HOFFMANN LA ROCHE (CH) 1999-06-02 CN disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed