SCHEMBL7702917

SCHEMBL7702917

Cc1ccc2c(c1)C(c1ccccn1)=NCC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.51
PARP1 P09874 1/20 0.41
PARP10 Q53GL7 1/20 0.41
PKM P14618 3/20 0.40
NPC1 O15118 3/20 0.40
KDM4E B2RXH2 3/20 0.40
RAB9A P51151 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
METAP1 P53582 2/20 0.39
METAP2 P50579 1/20 0.39
CBFB Q13951 1/20 0.39
MAPK10 P53779 1/20 0.38
GABRA1 P14867 2/20 0.38
GABRA5 P31644 2/20 0.38
GABRA3 P34903 2/20 0.38
GABRA2 P47869 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7701128 0.83 CYP1A2 (0.46) PARP1PARP10PKMNPC1KDM4E
SCHEMBL7702378 0.82 NPY5R (0.54) NPY5RPKMNPC1RAB9AALDH1A1
SCHEMBL7701012 0.82 NOS3 (0.49) NPY5RPKMNPC1KDM4ERAB9A
SCHEMBL28531265 0.79 MAPK10 (0.55) PKMALDH1A1MAPK10CHRM1LMNA
SCHEMBL30920956 0.77 CYP2A6 (0.40) NPY5RPKMNPC1KDM4ERAB9A
SCHEMBL4439294 0.74 MAPK10 (0.48) PARP1PARP10ALDH1A1MAPK10CYP19A1
SCHEMBL1009906 0.71 MAOA (0.53) NPY5RPARP1PARP10KDM4EALDH1A1
SCHEMBL3423163 0.71 KDM4E (0.50) NPY5RPKMNPC1KDM4ERAB9A
SCHEMBL29010811 0.71 MAPK10 (0.37) PARP1PARP10PKMALDH1A1MAPK10
SCHEMBL12164875 0.70 KDM4E (0.46) NPY5RPKMNPC1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed